SCHEMBL3619159

SCHEMBL3619159

Clc1cccc(-c2ccnc(NC3CCCCC3)n2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.59
PLK1 P53350 1/20 0.57
MAPK1 P28482 4/20 0.56
HDAC8 Q9BY41 1/20 0.56
HDAC6 Q9UBN7 1/20 0.56
IKBKB O14920 3/20 0.55
MAPK8 P45983 2/20 0.55
MAPK9 P45984 2/20 0.55
MAPK10 P53779 2/20 0.55
CNR2 P34972 1/20 0.54
EIF2AK2 P19525 1/20 0.54
CDC7 O00311 1/20 0.53
PLK4 O00444 1/20 0.53
JAK2 O60674 1/20 0.53
CCNB2 O95067 1/20 0.53
MAP4K4 O95819 1/20 0.53
INSR P06213 1/20 0.53
CDK1 P06493 1/20 0.53
CSF1R P07333 1/20 0.53
PIM1 P11309 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1030530 1.00 ADORA1 (0.59) ADORA1PLK1MAPK1HDAC8HDAC6
SCHEMBL1033923 0.88 IKBKB (0.59) ADORA1IKBKBMAPK8MAPK9MAPK10
SCHEMBL3653069 0.88 PLK1 (0.55) ADORA1PLK1MAPK1HDAC8HDAC6
SCHEMBL5819449 0.85 ADORA1 (0.52) ADORA1PLK1MAPK1HDAC8HDAC6
SCHEMBL1028968 0.85 MAP4K4 (0.55) MAPK1IKBKBMAPK8MAPK9MAPK10
SCHEMBL1033626 0.85 CDK1 (0.53) MAPK1IKBKBMAPK8MAPK9MAPK10
SCHEMBL1032138 0.84 IKBKB (0.76) MAPK1HDAC8HDAC6IKBKBMAPK8
SCHEMBL5823374 0.83 ADORA1 (0.53) ADORA1PLK1MAPK1HDAC8HDAC6
SCHEMBL5815500 0.83 TGFBR1 (0.54) ADORA1PLK1MAPK1HDAC8HDAC6
SCHEMBL2389822 0.83 IKBKB (0.55) PLK1MAPK1IKBKBMAPK8MAPK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010151747-A1 PYRIMINE COMPOUNDS AND METHODS OF MAKING AND USING SAME CYSTIC FIBROSIS FOUNDATION THERAPEUTICS, INC. (US) 2010-12-29 WO disclosed