SCHEMBL362463

SCHEMBL362463

CC(C=O)CN1CC(Oc2nc3c(N4CCOCC4)nc(Cl)nc3n2C)C1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 10/20 0.44
HDAC1 Q13547 1/20 0.40
TNF P01375 1/20 0.35
NT5E P21589 2/20 0.34
HRH3 Q9Y5N1 2/20 0.33
CYP3A4 P08684 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PIK3CA P42336 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL357452 0.80 PIK3CD (0.61) PIK3CDHDAC1TNFNT5ESMN1; SMN2
SCHEMBL362572 0.80 PIK3CD (0.42) PIK3CDHDAC1TNFNT5EHRH3
SCHEMBL370831 0.80 PIK3CD (0.60) PIK3CDPIK3CA
SCHEMBL18032516 0.79 TNF (0.42) PIK3CDHDAC1TNFNT5EHRH3
SCHEMBL369833 0.78 PIK3CD (0.75) PIK3CDPIK3CA
SCHEMBL371276 0.78 PIK3CD (0.49) PIK3CDTNFCYP3A4PIK3CA
SCHEMBL18032512 0.77 HDAC1 (0.42) PIK3CDHDAC1TNFNT5EHRH3
SCHEMBL18032511 0.76 PIK3CD (0.52) PIK3CDHDAC1TNFNT5EHRH3
SCHEMBL18032506 0.76 TNF (0.41) PIK3CDHDAC1TNFNT5EHRH3
SCHEMBL358553 0.75 PIK3CD (0.46) PIK3CDHDAC1TNFSMN1; SMN2PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593455-A1 PURINE COMPOUNDS SELECTIVE FOR I3 P110 DELTA, AND METHODS OF USE F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007493-A1 PURINE COMPOUNDS SELECTIVE FOR ΡI3Κ P110 DELTA, AND METHODS OF USE F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed