SCHEMBL3628534

SCHEMBL3628534

O=C1Oc2ccccc2CN1C1CCCNC1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.50
HTR2B P41595 11/20 0.41
HTR2C P28335 10/20 0.41
HTR2A P28223 3/20 0.39
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
HTR3A P46098 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
HTR3D Q70Z44 1/20 0.39
HTR3C Q8WXA8 1/20 0.39
MAPK1 P28482 1/20 0.36
HTR6 P50406 1/20 0.36
CAMK2D Q13557 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7400974 0.85 PARP1 (0.47) PARP1HTR2BHTR2CHTR2A
Hydrochloric Acid SCHEMBL11101784 0.83 PARP1 (0.46) PARP1HTR2BHTR2CHTR2A
SCHEMBL2784144 0.83 POLB (0.44) PARP1MAPK1
SCHEMBL21614132 0.77 PARP1 (0.59) PARP1HTR2BHTR2CHTR2AHTR3E
SCHEMBL30366187 0.77 PARP1 (0.59) PARP1HTR2BHTR2CHTR2AHTR3E
SCHEMBL31227444 0.70 PARP1 (0.45) PARP1HTR2BHTR2CHTR2AHTR3E
SCHEMBL31246891 0.70 PARP1 (0.45) PARP1HTR2BHTR2CHTR2AHTR3E
Hydrochloric Acid SCHEMBL7496829 0.70 HTR2C (0.47) PARP1HTR2BHTR2CHTR2A
Hydrochloric Acid SCHEMBL7400024 0.70 PARP1 (0.35) PARP1
SCHEMBL20986525 0.70 PARP1 (0.55) PARP1HTR2BHTR2CHTR2AHTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7795251-B2 3,4-dihydro-benzo[e][1,3]oxazin-2-ones NOVARTIS AG (CH) 2010-09-14 US disclosed
EP-1874742-A1 3,4-DIHYDRO-BENZO[E][1,3]OXAZIN-2-ONES Novartis AG (CH) 2008-01-09 EP disclosed
WO-2006108671-A1 3,4-DIHYDRO-BENZO[E][1,3]OXAZIN-2-ONES NOVARTIS AG (CH) 2006-10-19 WO disclosed