SCHEMBL362901

SCHEMBL362901

Cc1cc(Br)nc2ccccc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.64
BACE1 P56817 1/20 0.60
KDM4E B2RXH2 5/20 0.51
L3MBTL1 Q9Y468 3/20 0.51
MAPT P10636 3/20 0.51
POLB P06746 1/20 0.51
RAB9A P51151 1/20 0.51
GAA P10253 4/20 0.50
ALDH1A1 P00352 3/20 0.50
NPFFR1 Q9GZQ6 1/20 0.50
NPFFR2 Q9Y5X5 1/20 0.50
SMN1; SMN2 Q16637 3/20 0.49
HPGD P15428 2/20 0.49
ACHE P22303 1/20 0.49
KMT2A Q03164 2/20 0.47
LMNA P02545 2/20 0.47
TP53 P04637 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
GPR3 P46089 1/20 0.47
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29502790 0.78 CYP1A2 (1.00) CYP1A2BACE1KDM4EL3MBTL1MAPT
SCHEMBL29726892 0.78 BACE1 (0.44) CYP1A2BACE1KDM4EMAPTPOLB
SCHEMBL89010 0.78 CYP1A2 (1.00) CYP1A2BACE1KDM4EL3MBTL1MAPT
SCHEMBL1088580 0.78 CYP1A2 (0.69) CYP1A2BACE1KDM4EL3MBTL1MAPT
SCHEMBL1257332 0.78 BACE1 (0.44) CYP1A2BACE1KDM4EMAPTPOLB
Bromide SCHEMBL9222732 0.78 ADORA2A (0.47) CYP1A2BACE1MAPTPOLBALDH1A1
SCHEMBL9724208 0.78 KMT2A (0.51) CYP1A2KDM4EL3MBTL1MAPTPOLB
Hydrochloric Acid SCHEMBL11674460 0.77 CYP1A2 (0.96) CYP1A2BACE1KDM4EL3MBTL1MAPT
SCHEMBL423891 0.76 L3MBTL1 (0.71) CYP1A2BACE1KDM4EL3MBTL1MAPT
SCHEMBL10336509 0.76 CYP1A2 (0.60) CYP1A2BACE1KDM4EL3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110272383-A 2- is alkylated 4- methylquinoline, derivative and its synthetic method 湘潭大学 2019-09-24 CN claimed
CN-110003103-A A kind of two area side's acid quinoline dye of near-infrared and preparation method thereof 南通大学 2019-07-12 CN claimed
CN-115925685-B Triheteroaryltertiary amine and synthesis method thereof 南昌大学 2023-05-16 CN disclosed
CN-115925685-A Tri-heteroaryl tertiary amine and synthesis method thereof 南昌大学 2023-04-07 CN disclosed
WO-2023020512-A1 SUBSTITUTED PYRIDINE ANALOGUE, PREPARATION METHOD THEREFOR, AND USE THEREOF AS AHR MODULATOR 成都奥睿药业有限公司 2023-02-23 WO disclosed
CN-108947898-B Organic photoelectric functional material and application thereof 南京工业大学 2021-11-05 CN disclosed
CN-106187873-B A kind of aryl amine alkyl oxygen class compound and preparation method thereof 宜春学院 2019-11-05 CN disclosed
CN-110272383-A 2- is alkylated 4- methylquinoline, derivative and its synthetic method 湘潭大学 2019-09-24 CN disclosed
CN-110003103-A A kind of two area side's acid quinoline dye of near-infrared and preparation method thereof 南通大学 2019-07-12 CN disclosed
CN-108947898-A Organic photoelectric functional material and application thereof 南京工业大学 2018-12-07 CN disclosed
CN-108771681-A As the compound of DNA-PK inhibitor and its eutectic of deuterated derivatives 沃泰克斯药物股份有限公司 2018-11-09 CN disclosed
CN-106187873-A A kind of aryl amine alkyl oxygen compounds and preparation method thereof 宜春学院 2016-12-07 CN disclosed
CN-105814036-A Co-crystals of (S) -N-methyl-8- (1- ((2 '-methyl- [4, 5' -bipyrimidin ] -6-yl) amino) propan-2-yl) quinoline-4-carboxamide and deuterated derivatives thereof as DNA-PK inhibitors 沃泰克斯药物股份有限公司 2016-07-27 CN disclosed
CN-105636958-A Dna-pk inhibitors VERTEX PHARMA 2016-06-01 CN disclosed
CN-103003290-B Metal complexes MERCK PATENT GMBH (DE) 2016-05-04 CN disclosed
US-9331290-B2 Metal complexes MERCK PATENT GMBH (DE) 2016-05-03 US disclosed
US-20130112920-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2013-05-09 US disclosed
WO-2012007086-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2012-01-19 WO disclosed
CN-100345852-C Quinolinyl-pyrrolopyrazoles LILLY CO ELI (US) 2007-10-31 CN disclosed
CN-1714090-A Quinolinyl-pyrrolopyrazoles LILLY CO ELI (US) 2005-12-28 CN disclosed