SCHEMBL3630664

SCHEMBL3630664

COC(=O)c1ccnc(N)c1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 5/20 0.51
KDM4E B2RXH2 5/20 0.51
ALDH1A1 P00352 4/20 0.51
GLA P06280 2/20 0.51
ABL1 P00519 1/20 0.47
ATR Q13535 1/20 0.47
HSD17B10 Q99714 3/20 0.44
CFTR P13569 1/20 0.44
PSMD14 O00487 1/20 0.43
ATM Q13315 2/20 0.41
MAPT P10636 2/20 0.41
HPGD P15428 2/20 0.41
TSHR P16473 2/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
NQO2 P16083 3/20 0.40
MAP2K1 Q02750 1/20 0.40
POLB P06746 1/20 0.40
SLC40A1 Q9NP59 1/20 0.39
ROCK1 Q13464 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1970174 0.82 ATR (0.56) GAAKDM4EALDH1A1GLAABL1
SCHEMBL18224721 0.82 KDM4E (0.54) GAAKDM4EALDH1A1GLAABL1
SCHEMBL22911139 0.82 NUDT1 (0.50) KDM4EALDH1A1HSD17B10MAPTHPGD
SCHEMBL21749959 0.81 KDM4E (0.53) GAAKDM4EALDH1A1GLAABL1
SCHEMBL3553958 0.81 KDM4E (0.53) GAAKDM4EALDH1A1GLAABL1
SCHEMBL23500690 0.81 ATR (0.48) GAAKDM4EALDH1A1GLAABL1
SCHEMBL4075916 0.79 ATR (0.47) GAAKDM4EALDH1A1GLAABL1
SCHEMBL31032953 0.79 KDM4E (0.51) GAAKDM4EALDH1A1GLAABL1
SCHEMBL23500830 0.79 ATR (0.50) GAAKDM4EALDH1A1GLAABL1
SCHEMBL3943083 0.79 ATR (0.54) GAAKDM4EALDH1A1GLAABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2231662-B1 8-ANILINOIMIDAZOPYRIDINES AND THEIR USE AS ANTI-CANCER AND/OR ANTI-INFLAMMATORY AGENTS GENENTECH INC (US) 2011-06-22 EP disclosed
EP-2144898-A2 HETEROCYCLIC HYDRAZIDE COMPOUND AND PESTICIDAL USE OF THE SAME Sumitomo Chemical Company, Limited (JP) 2010-01-20 EP disclosed
WO-2009085980-A1 8-ANILIN0IMIDAZ0PYRIDINES AND THEIR USE AS ANTI-CANCER AND/OR ANTI-INFLAMMATORY AGENTS GENENTECH, INC. (US) 2009-07-09 WO disclosed
WO-2008130021-A2 HETEROCYCLIC HYDRAZIDE COMPOUND AND PESTICIDAL USE OF THE SAME SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2008-10-30 WO disclosed