SCHEMBL363146

SCHEMBL363146

Cc1cc(C(CC=NO)(c2ccccc2)c2ccccc2)ccn1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
UHRF1 Q96T88 1/20 0.33
PDK2 Q15119 1/20 0.32
KCNQ2 O43526 1/20 0.32
KIF11 P52732 6/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
CYP2D6 P10635 1/20 0.32
KCNH2 Q12809 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
MAPK1 P28482 2/20 0.31
WNT3A P56704 2/20 0.31
CYP1A2 P05177 1/20 0.31
HIF1A Q16665 1/20 0.31
GPBAR1 Q8TDU6 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362361 0.90 GPBAR1 (0.31) KIF11GPBAR1
SCHEMBL364470 0.85 CYP19A1 (0.34) KIF11
SCHEMBL362227 0.84 EDNRB (0.33) KIF11CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL363962 0.81
SCHEMBL364581 0.81
SCHEMBL363845 0.80
SCHEMBL364800 0.79 PDK2 (0.30) PDK2
SCHEMBL364230 0.79
SCHEMBL363284 0.79 TRPV1 (0.31)
SCHEMBL362561 0.79 RAB9A (0.32) KIF11CYP2D6MEN1KMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed