SCHEMBL3633141

SCHEMBL3633141

COC(=O)c1c2cc(=O)cc(OC)c-2cn(-c2ccccc2)c1C

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.57
MEN1 O00255 3/20 0.57
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 2/20 0.41
LMNA P02545 2/20 0.41
FGFR1 P11362 2/20 0.41
SRC P12931 1/20 0.41
MAPT P10636 4/20 0.41
HPGD P15428 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
PKM P14618 1/20 0.41
ALOX15 P16050 1/20 0.41
CYP2C19 P33261 1/20 0.41
HSD17B10 Q99714 1/20 0.41
NR4A2 P43354 1/20 0.40
ATM Q13315 2/20 0.39
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3630831 0.90 MEN1 (0.47) KMT2AMEN1KDM4EALDH1A1LMNA
SCHEMBL3627344 0.86 MEN1 (0.57) KMT2AMEN1KDM4EALDH1A1LMNA
SCHEMBL3628254 0.86 MEN1 (0.57) KMT2AMEN1KDM4EALDH1A1LMNA
SCHEMBL3631876 0.82 KMT2A (0.53) KMT2AMEN1KDM4EALDH1A1LMNA
SCHEMBL28697581 0.79 MEN1 (0.69) KMT2AMEN1KDM4EALDH1A1LMNA
SCHEMBL28672791 0.77 MEN1 (0.61) KMT2AMEN1KDM4EALDH1A1LMNA
SCHEMBL3633407 0.76 PDE4D (0.46) KMT2AMEN1KDM4EALDH1A1MAPT
SCHEMBL3632614 0.75 MEN1 (0.45) KMT2AMEN1KDM4EALDH1A1MAPT
SCHEMBL3628896 0.74 ALDH1A1 (0.45) KMT2AMEN1KDM4EALDH1A1MAPT
SCHEMBL28931713 0.74 MEN1 (0.58) KMT2AMEN1KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150534-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2010-02-10 EP disclosed
WO-2008131779-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2008-11-06 WO disclosed