SCHEMBL3635907

SCHEMBL3635907

Cc1cc(F)ccc1C(C(N)=O)N1CCN2CCC[C@@H]2C1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
NPC1 O15118 1/20 0.39
GHSR Q92847 1/20 0.38
DPP4 P27487 4/20 0.38
DPP9 Q86TI2 4/20 0.38
DPP7 Q9UHL4 4/20 0.38
DPP8 Q6V1X1 3/20 0.38
SIGMAR1 Q99720 1/20 0.38
GRM2 Q14416 1/20 0.37
TP53 P04637 1/20 0.37
POLB P06746 1/20 0.37
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3638555 0.85 CHRM2 (0.51) CHRM2CHRM1NPC1POLB
SCHEMBL13984260 0.83 MEN1 (0.38) NPC1DPP4DPP9DPP7DPP8
SCHEMBL3639687 0.80 KMT2A (0.41) CHRM2CHRM1GHSRPOLB
SCHEMBL3638732 0.79 GHSR (0.64) GHSRSIGMAR1
SCHEMBL3637111 0.78 TSHR (0.38) CHRM2CHRM1NPC1SIGMAR1POLB
SCHEMBL3636129 0.76 GHSR (0.45) CHRM2CHRM1GHSRTP53POLB
SCHEMBL13078460 0.74 GHSR (0.56) GHSR
SCHEMBL13044855 0.74 TSHR (0.42) CHRM1GHSRPOLB
Hydrochloric Acid SCHEMBL3638182 0.73 TSHR (0.41) CHRM1GHSRPOLB
Hydrochloric Acid SCHEMBL3742803 0.73 TSHR (0.41) CHRM1GHSRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100286152-A1 N-PHENYL HYDRAZIDES AS MODULATORS OF THE GHRELIN RECEPTOR GLAXO GROUP LIMITED (GB) 2010-11-11 US disclosed
US-20100286152-A1 N-PHENYL HYDRAZIDES AS MODULATORS OF THE GHRELIN RECEPTOR GLAXO GROUP LIMITED (GB) 2010-11-11 US disclosed
US-20100286152-A1 N-PHENYL HYDRAZIDES AS MODULATORS OF THE GHRELIN RECEPTOR GLAXO GROUP LIMITED (GB) 2010-11-11 US disclosed
EP-2167466-A1 N-PHENYL HYDRAZIDES AS MODULATORS OF THE GHRELIN RECEPTOR Glaxo Group Limited (GB) 2010-03-31 EP disclosed
WO-2008148853-A1 N-PHENYL HYDRAZIDES AS MODULATORS OF THE GHRELIN RECEPTOR GLAXO GROUP LIMITED (GB) 2008-12-11 WO disclosed
WO-2008148853-A1 N-PHENYL HYDRAZIDES AS MODULATORS OF THE GHRELIN RECEPTOR GLAXO GROUP LIMITED (GB) 2008-12-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100286152-A1 N-PHENYL HYDRAZIDES AS MODULATORS OF THE GHRELIN RECEPTOR GIPR, GHSR, GLP1R CHRM2 1777/4885CHRM1 1896/4885NPC1 975/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.