SCHEMBL3636175

SCHEMBL3636175

Cc1ccc(-c2nc(NN3C(=O)CC(C)(C)C3=O)ccc2C(F)(F)F)cc1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
XPO1 O14980 12/20 0.40
AR P10275 1/20 0.37
TRPV1 Q8NER1 2/20 0.35
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
KDM1A O60341 1/20 0.31
PTGS2 P35354 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GLA P06280 1/20 0.30
GAA P10253 1/20 0.30
HPGD P15428 1/20 0.30
ATM Q13315 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1593000 0.80 XPO1 (0.48) XPO1TRPV1CYP11B1CYP11B2PTGS2
SCHEMBL1593002 0.78 XPO1 (0.44) XPO1TRPV1CYP11B1CYP11B2KDM1A
SCHEMBL1592494 0.71 XPO1 (0.51) XPO1PTGS2
SCHEMBL1592486 0.71 XPO1 (0.48) XPO1ALDH1A1
SCHEMBL30176895 0.69 XPO1 (0.34) XPO1TRPV1CYP11B1CYP11B2
SCHEMBL30346302 0.68 XPO1 (0.63) XPO1TRPV1CYP11B2GAA
SCHEMBL1592487 0.68 XPO1 (0.43) XPO1TRPV1
SCHEMBL1592440 0.65 XPO1 (0.47) XPO1
SCHEMBL1592800 0.64 XPO1 (0.48) XPO1PTGS2
SCHEMBL20880362 0.62 XPO1 (0.54) XPO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2152692-A2 COMPOUNDS WITH ANTI-CANCER ACTIVITY Canbas Co. Ltd. (JP) 2010-02-17 EP claimed
WO-2009031040-A2 COMPOUNDS WITH ANTI-CANCER ACTIVITY CANBAS CO., LTD. (JP) 2009-03-12 WO claimed