SCHEMBL3636435

SCHEMBL3636435

CCCc1nc2c(C)cc(C(=O)N(CCS)C(I)c3ccccc3)cc2n1Cc1ccc(C(=O)O)cc1

nearest known ligand 0.54

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 19/20 0.54
AGTR2 P50052 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Toluene SCHEMBL16460869 0.80 AGTR1 (0.59) AGTR1AGTR2
SCHEMBL3640166 0.79 PPARG (0.68) AGTR1
SCHEMBL3637893 0.76 AGTR1 (0.65) AGTR1AGTR2
SCHEMBL4887978 0.76 AGTR1 (0.60) AGTR1AGTR2
SCHEMBL4884086 0.76 AGTR1 (0.51) AGTR1AGTR2
SCHEMBL4880144 0.73 AGTR1 (0.59) AGTR1AGTR2
SCHEMBL29387259 0.73 AGTR1 (0.82) AGTR1AGTR2
SCHEMBL8266757 0.73 AGTR1 (0.82) AGTR1AGTR2
SCHEMBL4887839 0.72 AGTR1 (0.57) AGTR1AGTR2
SCHEMBL4887823 0.72 AGTR1 (0.57) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2162442-A1 DUAL-ACTING BENZOIMIDAZOLE ANTIHYPERTENSIVE AGENTS Theravance, Inc. (US) 2010-03-17 EP disclosed
WO-2008153857-A1 DUAL-ACTING BENZOIMIDAZOLE ANTIHYPERTENSIVE AGENTS THERAVANCE, INC. (US) 2008-12-18 WO disclosed