SCHEMBL3636602

SCHEMBL3636602

O=C(O)C1C=CC=CC1(F)Nc1ccccc1

nearest known ligand 0.32

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 2/20 0.32
EPHX2 P34913 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
TP53 P04637 1/20 0.32
TSHR P16473 1/20 0.32
CDK9 P50750 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
NAPRT Q6XQN6 1/20 0.31
HSD17B10 Q99714 1/20 0.31
POLB P06746 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
RAB9A P51151 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
GAA P10253 2/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30870483 0.78 TP53 (0.32) EPHX1EPHX2SMN1; SMN2TP53TSHR
SCHEMBL11163620 0.78 NAPRT (0.34) EPHX1EPHX2SMN1; SMN2TP53TSHR
SCHEMBL11584096 0.76 TSHR (0.38) EPHX1EPHX2SMN1; SMN2TP53TSHR
SCHEMBL5391078 0.71
SCHEMBL3267769 0.71 KCNJ6 (0.32) MEN1KMT2A
SCHEMBL4216034 0.70 HSD11B1 (0.38) SMN1; SMN2TSHRHSD17B10MEN1KMT2A
SCHEMBL8343262 0.70 TSHR (0.40) EPHX1EPHX2SMN1; SMN2TP53TSHR
SCHEMBL574722 0.67 HSD11B1 (0.36) LMNA
SCHEMBL5789431 0.66
SCHEMBL8543332 0.66 PTPN1 (0.36) SMN1; SMN2TSHRHSD17B10TDP1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2148862-A1 DIHYDROQUINONE AND DIHYDRONAPHTHRIDINE INHIBITORS OF JNK F. Hoffmann-Roche AG (CH) 2010-02-03 EP disclosed
WO-2008138920-A1 DIHYDROQUINONE AND DIHYDRONAPHTHRIDINE INHIBITORS OF JNK F. HOFFMANN-LA ROCHE AG (CH) 2008-11-20 WO disclosed