SCHEMBL3638680

SCHEMBL3638680

C[C@]1(c2ccccc2)CCN(c2cccc(-c3cccc(Cl)c3)c2)C(=O)O1

nearest known ligand 0.89

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 17/20 0.89
CYP2C9 P11712 1/20 0.44
BACE1 P56817 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL958988 1.00 HSD11B1 (0.89) HSD11B1CYP2C9BACE1
SCHEMBL957964 0.94 HSD11B1 (0.83) HSD11B1CYP2C9
SCHEMBL3644262 0.94 HSD11B1 (0.83) HSD11B1CYP2C9
SCHEMBL958989 0.94 HSD11B1 (1.00) HSD11B1CYP2C9
SCHEMBL3643940 0.92 HSD11B1 (1.00) HSD11B1CYP2C9
SCHEMBL957231 0.92 HSD11B1 (1.00) HSD11B1CYP2C9
SCHEMBL955206 0.88 HSD11B1 (0.79) HSD11B1CYP2C9
SCHEMBL957986 0.87 HSD11B1 (0.86) HSD11B1CYP2C9
SCHEMBL3639706 0.87 HSD11B1 (0.77) HSD11B1CYP2C9
SCHEMBL956746 0.87 HSD11B1 (0.77) HSD11B1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2183228-A1 CYCLIC INHIBITORS OF 11ß -HYDROXYSTERIOD DEHYDROGENASE 1 Vitae Pharmaceuticals, Inc. (US) 2010-05-12 EP claimed
WO-2009017664-A1 CYCLIC INHIBITORS OF 11β-HYDROXYSTERIOD DEHYDROGENASE 1 VITAE PHARMACEUTICALS, INC. (US) 2009-02-05 WO claimed