SCHEMBL3638870

SCHEMBL3638870

CC(C)(C)C(=O)N1CCN(c2nc(NCc3ccccc3)c3ccccc3n2)CC1.CC(C)C(=O)N1CCN(c2nc(NCc3ccccc3)c3ccccc3n2)CC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 4/20 0.60
PDE5A O76074 2/20 0.60
HTR2A P28223 1/20 0.56
DRD3 P35462 1/20 0.56
KDM4E B2RXH2 3/20 0.56
MAPT P10636 2/20 0.56
NPSR1 Q6W5P4 2/20 0.56
MAPK1 P28482 1/20 0.56
CTNNB1 P35222 6/20 0.52
TCF7L2 Q9NQB0 6/20 0.52
HTR3A P46098 1/20 0.48
ALOX15 P16050 1/20 0.46
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
HTT P42858 1/20 0.45
KMT2A Q03164 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
MCHR1 Q99705 1/20 0.44
APP P05067 1/20 0.44
ACHE P22303 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3640608 0.93 HRH4 (0.69) HRH4PDE5AHTR2ADRD3KDM4E
SCHEMBL3638488 0.93 HRH4 (0.69) HRH4PDE5AHTR2ADRD3KDM4E
SCHEMBL3641800 0.82 HRH4 (0.72) HRH4PDE5AHTR2ADRD3KDM4E
SCHEMBL13009783 0.81 ACHE (0.66) HRH4PDE5AHTR2ADRD3KDM4E
SCHEMBL3640288 0.79 PDE5A (0.68) HRH4PDE5AHTR2ADRD3KDM4E
SCHEMBL3644233 0.78 PDE5A (0.67) HRH4PDE5AHTR2ADRD3KDM4E
SCHEMBL3640234 0.76 HRH4 (1.00) HRH4PDE5AHTR2ADRD3KDM4E
SCHEMBL27808528 0.75 CTNNB1 (0.68) HRH4PDE5AHTR2ADRD3KDM4E
Hydrochloric Acid SCHEMBL3637430 0.75 HRH4 (0.97) HRH4PDE5AHTR2ADRD3KDM4E
SCHEMBL2628837 0.75 PDE5A (0.79) HRH4PDE5AHTR2ADRD3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2173346-A2 USE OF COMPOUNDS FOR PREPARING ANTI-TUBERCULOSIS AGENTS Summit Corporation Plc (GB) 2010-04-14 EP disclosed
WO-2009001060-A2 USE OF COMPOUNDS FOR PREPARING ANTI-TUBERCULOSIS AGENTS SUMMIT CORPORATION PLC (GB) 2008-12-31 WO disclosed