SCHEMBL3645569

SCHEMBL3645569

CNC(=O)c1cccc(-c2cn[nH]c(=O)c2)c1.CNC(=O)c1cccc(C2=CC(Cl)NN=C2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 1/20 0.43
CRBN Q96SW2 1/20 0.38
CYP17A1 P05093 1/20 0.36
CYP3A4 P08684 1/20 0.36
ROCK2 O75116 2/20 0.35
ROCK1 Q13464 1/20 0.35
CDK7 P50613 1/20 0.35
MEN1 O00255 1/20 0.35
OPRK1 P41145 1/20 0.35
KMT2A Q03164 1/20 0.35
NR4A2 P43354 1/20 0.35
TNIK Q9UKE5 1/20 0.35
PDK2 Q15119 1/20 0.34
BRD4 O60885 1/20 0.34
CREBBP Q92793 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
TAF1 P21675 1/20 0.34
FGFR1 P11362 1/20 0.34
FGFR3 P22607 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL836826 0.83 CDK8 (0.57) CDK8CRBNCYP17A1CYP3A4ROCK2
SCHEMBL3645370 0.79 CDK8 (0.51) CDK8CRBNCYP17A1CYP3A4ROCK2
SCHEMBL836582 0.74 CDK8 (0.44) CDK8CRBNCYP17A1CYP3A4NR4A2
SCHEMBL9949385 0.69 CDK8 (0.57) CDK8PDK2
SCHEMBL13702375 0.67 HDAC8 (0.68) CDK8CRBNCYP17A1CYP3A4NR4A2
SCHEMBL12319279 0.64 PLK1 (0.39) CDK8ROCK2LRRK2
SCHEMBL13702359 0.63 CRBN (0.56) CDK8CRBNCYP17A1CYP3A4ROCK2
SCHEMBL723332 0.63 HDAC8 (0.70) CDK8CRBNPDK2
SCHEMBL10538440 0.62 NOTUM (0.49) BRD4
SCHEMBL5562512 0.62 NOTUM (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2183027-A1 ORGANIC COMPOUNDS Novartis Ag (CH) 2010-05-12 EP disclosed
WO-2009013335-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2009-01-29 WO disclosed