SCHEMBL3645370

SCHEMBL3645370

CNC(=O)c1cccc(-c2cn[nH]c(=O)c2)c1.O=c1cc(Cl)cn[nH]1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 1/20 0.51
NR4A2 P43354 1/20 0.45
CRBN Q96SW2 1/20 0.45
ROCK2 O75116 3/20 0.44
ROCK1 Q13464 1/20 0.44
CDK7 P50613 1/20 0.43
PDK2 Q15119 1/20 0.42
CYP17A1 P05093 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAOA P21397 2/20 0.41
MAOB P27338 2/20 0.41
LRRK2 Q5S007 1/20 0.41
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
CSNK1D P48730 1/20 0.40
BRD4 O60885 1/20 0.40
CREBBP Q92793 1/20 0.40
TNIK Q9UKE5 1/20 0.39
TAF1 P21675 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL836826 0.93 CDK8 (0.57) CDK8NR4A2CRBNROCK2ROCK1
SCHEMBL3645569 0.79 CDK8 (0.43) CDK8NR4A2CRBNROCK2ROCK1
SCHEMBL9949385 0.77 CDK8 (0.57) CDK8PDK2
SCHEMBL10538440 0.74 NOTUM (0.49) BRD4
SCHEMBL13702375 0.74 HDAC8 (0.68) CDK8NR4A2CRBNPDK2CYP17A1
SCHEMBL12319279 0.71 PLK1 (0.39) CDK8ROCK2LRRK2HDAC8HDAC6
SCHEMBL13702359 0.70 CRBN (0.56) CDK8NR4A2CRBNROCK2PDK2
SCHEMBL723332 0.70 HDAC8 (0.70) CDK8CRBNPDK2HDAC8HDAC6
SCHEMBL388422 0.69
SCHEMBL5562512 0.69 NOTUM (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2183027-A1 ORGANIC COMPOUNDS Novartis Ag (CH) 2010-05-12 EP disclosed
WO-2009013335-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2009-01-29 WO disclosed