Fluorouracil

Fluorouracil

SCHEMBL3646

O=c1[nH]cc(F)c(=O)[nH]1

nearest known ligand 0.00

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

TYMS

The experimentally established mechanism targets of Fluorouracil. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fluorouracil SCHEMBL10017187 1.00
Fluorouracil SCHEMBL249289 1.00 MAPT (1.00)
Fluorouracil SCHEMBL31441196 0.97 MAPT (0.95)
Fluorouracil SCHEMBL21880166 0.97 MAPT (0.95)
Fluorouracil SCHEMBL30439198 0.97 MAPT (0.95)
Fluorouracil SCHEMBL11327829 0.97 MAPT (0.95)
Fluorouracil SCHEMBL7650203 0.97 MAPT (0.95)
Fluorouracil SCHEMBL21527805 0.97 MAPT (0.95)
Fluorouracil SCHEMBL15284932 0.97 MAPT (0.95)
Fluorouracil SCHEMBL28803776 0.97 MAPT (0.95)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 331336 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12186394-B2 Compositions and methods for treatment of pre-cancerous skin lesions WASHINGTON UNIVERSITY (US) 2025-01-07 US claimed
US-12187782-B2 PDL1 peptides for use in cancer vaccines IO BIOTECH APS (DK) 2025-01-07 US claimed
EP-4484420-A1 INHIBITOR OF INTERACTION BETWEEN YAP/TAZ AND TEAD, PREPARATION THEREOF, PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF Etern Biopharma (Shanghai) Co., Ltd. (CN) 2025-01-01 EP claimed
CN-119185165-A Controlled release medicine micro-needle with good biocompatibility and preparation method thereof 上海市第一人民医院 2024-12-27 CN claimed
CN-119191955-A Enantiomer-eudesmane sesquiterpenoids and application thereof 海南师范大学 2024-12-27 CN claimed
US-20240425752-A1 BILIRUBIN-COATED RADIO-LUMINESCENT PARTICLES PURDUE RESEARCH FOUNDATION (US) 2024-12-26 US claimed
US-20240423972-A1 CHEMOTHERAPEUTIC BIOADHESIVE PARTICLES WITH IMMUNOSTIMULATORY MOLECULES FOR CANCER TREATMENT YALE UNIVERSITY 2024-12-26 US claimed
EP-4479034-A1 CAPSAICIN DERIVATIVES AS BIOENHANCERS ON ACTIVE SUBSTANCES METABOLIZED BY CYP1A2 AND CYP2D6 aXichem AB (SE) 2024-12-25 EP claimed
US-12173039-B1 TPL2 inhibiting agents, uses thereof, and detection of TPL2 WASHINGTON UNIVERSITY (US) 2024-12-24 US claimed
US-20240415972-A1 MICROFRAGMENTED FAT TISSUE AS DRUG DELIVERY SYSTEM IN LIVER CANCER THERAPY LIPOGEMS INT S P A (IT) 2024-12-19 US claimed
US-3992522-A INFLUENZA VIRUSES THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH, EDUCATION AND WELFARE (US) 1976-11-16 US claimed
US-3992208-A Photo-sensitive etchant and method for forming metal image using same FUJI PHOTO FILM CO., LTD. (JA) 1976-11-16 US claimed
US-3991203-A Vehicle composition containing 1-substituted azacyclopentan-2-ones NELSON RESEARCH & DEVELOPMENT COMPANY (US) 1976-11-09 US claimed
US-3989815-A PENETRATION OF SKINS NELSON RESEARCH & DEVELOPMENT COMPANY (US) 1976-11-02 US claimed
US-3989816-A PENETRATION OF SKINS OR MEMBRANES NELSON RESEARCH & DEVELOPMENT COMPANY (US) 1976-11-02 US claimed
US-3971784-A ANTIMETABOLITES MITSUI PHARMACEUTICALS, INCORPORATED (JA) 1976-07-27 US claimed
US-3966924-A B-METHASONE VALERATE, 5-FLUOROURACIL ALLERGAN PHARMACEUTICALS (US) 1976-06-29 US claimed
US-3960864-A Method of synthesizing 1-(tetrahydro-2-furanyl)-5-fluorouracil THE UNIVERSITY OF UTAH (US) 1976-06-01 US claimed
US-3954536-A 5-FLUORO-URACIL, GLUCOSE, GLYCERIN LIQUICHIMICA S.P.A. (IT) 1976-05-04 US claimed
US-3954758-A GERMICIDES, CANCER CHEMOTHERAPY PCR, INC. (US) 1976-05-04 US claimed