SCHEMBL365095

SCHEMBL365095

Cc1ccc(/C(CC(c2ccc(-c3ccc(C(=O)O)c(F)c3)cc2)c2ccc(Cl)cc2Cl)=N/O)[nH]c1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.37
ADRB1 P08588 4/20 0.36
ADRB3 P13945 4/20 0.36
RARB P10826 3/20 0.33
RARA P10276 2/20 0.33
F9 P00740 2/20 0.33
RARG P13631 1/20 0.33
FFAR1 O14842 1/20 0.33
ADRA2A P08913 1/20 0.33
CLCN2 P51788 1/20 0.33
HAO1 Q9UJM8 1/20 0.32
DHODH Q02127 1/20 0.31
PLA2G4A P47712 1/20 0.31
MRGPRX4 Q96LA9 1/20 0.31
TSHR P16473 1/20 0.30
CASP1 P29466 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
SLC1A3 P43003 1/20 0.30
SLC1A2 P43004 1/20 0.30
SLC1A1 P43005 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363296 0.85 GPBAR1 (0.38) GPBAR1ADRB1ADRB3RARBRARA
SCHEMBL362646 0.85 GPBAR1 (0.38) GPBAR1ADRB1ADRB3RARBRARA
SCHEMBL363787 0.85 GPBAR1 (0.38) GPBAR1ADRB1ADRB3RARBRARA
SCHEMBL1389726 0.79 GPBAR1 (0.37) GPBAR1ADRB1ADRB3RARBRARA
SCHEMBL1389759 0.79 GPBAR1 (0.37) GPBAR1ADRB1ADRB3RARBRARA
SCHEMBL1389965 0.79 GPBAR1 (0.37) GPBAR1ADRB1ADRB3RARBRARA
SCHEMBL1389729 0.79 GPBAR1 (0.37) GPBAR1ADRB1ADRB3RARBRARA
SCHEMBL1389761 0.79 GPBAR1 (0.37) GPBAR1ADRB1ADRB3RARBRARA
SCHEMBL1389964 0.79 GPBAR1 (0.37) GPBAR1ADRB1ADRB3RARBRARA
SCHEMBL1389961 0.79 GPBAR1 (0.37) GPBAR1ADRB1ADRB3RARBRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed