SCHEMBL363296

SCHEMBL363296

Cc1cc(/C(CC(c2ccc(-c3ccc(C(=O)O)c(F)c3)cc2)c2ccc(Cl)cc2Cl)=N/O)c[nH]c1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.38
ADRB1 P08588 4/20 0.35
ADRB3 P13945 4/20 0.35
RARB P10826 3/20 0.33
RARA P10276 2/20 0.33
MGAM O43451 1/20 0.33
GAA P10253 1/20 0.33
SI P14410 1/20 0.33
MGAM2 Q2M2H8 1/20 0.33
RARG P13631 1/20 0.33
FFAR1 O14842 1/20 0.33
ERCC1 P07992 1/20 0.32
ERCC4 Q92889 1/20 0.32
PRKAB2 O43741 2/20 0.32
PRKAG1 P54619 2/20 0.32
PRKAA2 P54646 2/20 0.32
PRKAA1 Q13131 2/20 0.32
PRKAG3 Q9UGI9 2/20 0.32
PRKAG2 Q9UGJ0 2/20 0.32
PRKAB1 Q9Y478 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363787 1.00 GPBAR1 (0.38) GPBAR1ADRB1ADRB3RARBRARA
SCHEMBL362646 1.00 GPBAR1 (0.38) GPBAR1ADRB1ADRB3RARBRARA
SCHEMBL364998 0.94 GPBAR1 (0.39) GPBAR1ADRB1ADRB3RARBRARA
SCHEMBL363089 0.94 GPBAR1 (0.39) GPBAR1ADRB1ADRB3RARBRARA
SCHEMBL364367 0.94 GPBAR1 (0.39) GPBAR1ADRB1ADRB3RARBRARA
SCHEMBL361844 0.91 GPBAR1 (0.44) GPBAR1ADRB1ADRB3RARBRARA
SCHEMBL362317 0.87 GPBAR1 (0.52) GPBAR1ADRB1ADRB3RARBRARA
SCHEMBL361680 0.86 GPBAR1 (0.47) GPBAR1ADRB1ADRB3MGAMGAA
SCHEMBL365095 0.85 GPBAR1 (0.37) GPBAR1ADRB1ADRB3RARBRARA
SCHEMBL363679 0.84 GPBAR1 (0.42) GPBAR1ADRB1ADRB3RARBMGAM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed