SCHEMBL365142

SCHEMBL365142

C/C=C/c1ccc(OC)c(N)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 3/20 0.71
TUBB1 Q9H4B7 5/20 0.67
TUBB4A P04350 4/20 0.67
TUBB P07437 4/20 0.67
TUBA3C P0DPH7 4/20 0.67
TUBA1B P68363 4/20 0.67
TUBA4A P68366 4/20 0.67
TUBB4B P68371 4/20 0.67
TUBB3 Q13509 4/20 0.67
TUBB2A Q13885 4/20 0.67
TUBB8 Q3ZCM7 4/20 0.67
TUBA3E Q6PEY2 4/20 0.67
TUBA1A Q71U36 4/20 0.67
TUBA1C Q9BQE3 4/20 0.67
TUBB6 Q9BUF5 4/20 0.67
TUBB2B Q9BVA1 4/20 0.67
TYR P14679 1/20 0.58
CYP19A1 P11511 1/20 0.53
ALDH1A1 P00352 3/20 0.52
CYP3A4 P08684 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25990122 0.85 APP (0.71) APPTUBB1TUBB4ATUBBTUBA3C
Methylisoeugenol SCHEMBL112937 0.82 TYR (0.69) APPTUBB1TUBB4ATUBBTUBA3C
Methylisoeugenol SCHEMBL29518298 0.82 TYR (0.69) APPTUBB1TUBB4ATUBBTUBA3C
Methylisoeugenol SCHEMBL1760676 0.82 TYR (0.69) APPTUBB1TUBB4ATUBBTUBA3C
Methylisoeugenol SCHEMBL30203196 0.82 TYR (0.69) APPTUBB1TUBB4ATUBBTUBA3C
Methylisoeugenol SCHEMBL1532669 0.82 TYR (0.69) APPTUBB1TUBB4ATUBBTUBA3C
Methylisoeugenol SCHEMBL29364555 0.82 TYR (0.69) APPTUBB1TUBB4ATUBBTUBA3C
SCHEMBL291904 0.80 TUBB1 (1.00) APPTUBB1TUBB4ATUBBTUBA3C
SCHEMBL13660060 0.80 TUBB1 (0.76) APPTUBB1TUBB4ATUBBTUBA3C
SCHEMBL1284983 0.80 NQO2 (0.72) APPTUBB1TUBB4ATUBBTUBA3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593457-A1 PYRAZOLO [1, 5A]PYRIMIDINE AND THIENO [3, 2B]PYRIMIDINE DERIVATIVES AS IRAK4 MODULATORS F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007375-A1 PYRAZOLO [1, 5A] PYRIMIDINE AND THIENO [3, 2B] PYRIMIDINE DERIVATIVES AS IRAK4 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed