SCHEMBL3651908

SCHEMBL3651908

CC(C)(C)Cc1nc(-c2ccccc2F)c(Sc2ccccc2)s1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
POLB P06746 1/20 0.35
ALDH1A1 P00352 5/20 0.34
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HTR3A P46098 1/20 0.33
ADORA2A P29274 1/20 0.33
MBNL1 Q9NR56 1/20 0.33
MPL P40238 1/20 0.32
DPP4 P27487 1/20 0.32
CNR2 P34972 1/20 0.31
DCUN1D1 Q96GG9 1/20 0.31
ADORA2B P29275 1/20 0.30
ADORA1 P30542 1/20 0.30
APEX1 P27695 1/20 0.30
GRM2 Q14416 1/20 0.30
FBP1 P09467 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2844203 0.83 DPP4 (0.41) MAPTNPC1RAB9AALDH1A1GAA
SCHEMBL3650619 0.81 ALDH1A1 (0.32) MAPTNPC1RAB9APOLBALDH1A1
SCHEMBL3654417 0.80 MEN1 (0.33) MAPTNPC1RAB9AALDH1A1GAA
SCHEMBL4129352 0.80 MAPT (0.35) MAPTNPC1RAB9AALDH1A1GAA
SCHEMBL4125425 0.78 ALDH1A1 (0.36) MAPTNPC1RAB9APOLBALDH1A1
SCHEMBL3650614 0.78 CTSA (0.34) MAPTALDH1A1SMN1; SMN2
SCHEMBL3650616 0.77 HTR2C (0.37)
SCHEMBL3696085 0.70 MAP4K1 (0.32) POLBALDH1A1SMN1; SMN2L3MBTL1KDM4E
SCHEMBL3652892 0.70 PPARG (0.33)
SCHEMBL3807952 0.69 MAPT (0.33) MAPTALDH1A1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed