SCHEMBL3652964

SCHEMBL3652964

CC(C)(C)OC(=O)N1CCC(=O)C(Br)C1.CC(C)(C)OC(=O)N1CCC(=O)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
EPHX1 P07099 1/20 0.41
MAPT P10636 2/20 0.40
KDM4E B2RXH2 1/20 0.40
THRB P10828 1/20 0.40
DDB1 Q16531 2/20 0.40
CRBN Q96SW2 2/20 0.40
HPGD P15428 1/20 0.40
GPR119 Q8TDV5 3/20 0.39
ESR2 Q92731 1/20 0.39
ELANE P08246 1/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
RECQL P46063 1/20 0.38
NR1H2 P55055 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL166445 0.94 USP2 (0.42) USP2SMN1; SMN2EPHX1MAPTKDM4E
SCHEMBL173426 0.86 HPGD (0.44) USP2SMN1; SMN2EPHX1MAPTKDM4E
SCHEMBL171462 0.84 EPHX1 (0.50) USP2SMN1; SMN2EPHX1MAPTKDM4E
SCHEMBL31028 0.83 USP2 (0.56) USP2SMN1; SMN2EPHX1MAPTKDM4E
SCHEMBL27669441 0.83 USP2 (0.56) USP2SMN1; SMN2EPHX1MAPTKDM4E
Ammonia Solution, Strong SCHEMBL27841683 0.82 USP2 (0.55) USP2SMN1; SMN2EPHX1MAPTKDM4E
Iodomethane SCHEMBL15848230 0.80 USP2 (0.53) USP2SMN1; SMN2EPHX1MAPTKDM4E
Ethylene SCHEMBL3832936 0.80 USP2 (0.53) USP2SMN1; SMN2EPHX1MAPTKDM4E
SCHEMBL26093324 0.79 NR1H2 (0.43) USP2SMN1; SMN2EPHX1MAPTKDM4E
SCHEMBL12908934 0.78 USP2 (0.44) USP2SMN1; SMN2EPHX1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197552-A2 NOVEL TETRAHYDROFUSEDPYRIDINES AS HISTONE DEACETYLASE INHIBITORS 4SC AG (DE) 2010-06-23 EP disclosed
WO-2009037001-A2 NOVEL TETRAHYDROFUSEDPYRIDINES AS HISTONE DEACETYLASE INHIBITORS 4SC AG (DE) 2009-03-26 WO disclosed