SCHEMBL3653705

SCHEMBL3653705

CC(C)(C)C(Cc1nc(-c2cccnc2F)c(Sc2ccnc(Cl)c2)s1)NC(=O)O

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.33
ROCK2 O75116 1/20 0.32
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
DYRK1A Q13627 1/20 0.32
LIPC P11150 1/20 0.31
LIPG Q9Y5X9 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
MAPK14 Q16539 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3650216 0.90 POLB (0.36) DHODHROCK2DYRK1AMAPK14
SCHEMBL3655560 0.89 DHODH (0.34) DHODHROCK2DYRK1AMAPK14
SCHEMBL3804237 0.85 DYRK1A (0.33) DHODHAKR1C3AKR1C2DYRK1ALIPC
SCHEMBL4123415 0.81 MAPK14 (0.34) DHODHROCK2DYRK1ALIPCLIPG
SCHEMBL4123409 0.81 DHODH (0.34) DHODHROCK2LIPCLIPGPTGDR2
SCHEMBL3653706 0.80 DHODH (0.32) DHODHROCK2PTGDR2
SCHEMBL3652261 0.79 DHODH (0.35) DHODHROCK2DYRK1ALIPCLIPG
SCHEMBL3651371 0.79 CTSA (0.33)
SCHEMBL3650614 0.78 CTSA (0.34)
SCHEMBL3652596 0.78 CACNA1G (0.34) ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed