SCHEMBL3655147

SCHEMBL3655147

CC(C)CCCNc1ccc(C(F)(F)F)cc1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.43
ALDH1A1 P00352 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
RHOC P08134 2/20 0.40
RHOA P61586 2/20 0.40
EPHX2 P34913 1/20 0.39
CDK1 P06493 1/20 0.38
FFAR1 O14842 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
MMP2 P08253 1/20 0.38
ADRA2A P08913 1/20 0.37
CACNA1B Q00975 1/20 0.37
HDAC1 Q13547 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3657741 0.82 XPO1 (0.43) ALDH1A1LMNARHOCRHOAADRA2A
SCHEMBL19314147 0.79 MAPT (0.61) ALDH1A1MEN1KMT2AHTTSMN1; SMN2
SCHEMBL8178051 0.79 MEN1 (0.61) KIF11MEN1KMT2ALMNAHTT
SCHEMBL9515478 0.79 PRSS1 (0.46) ALDH1A1MEN1KMT2ALMNAHTT
SCHEMBL19669164 0.78 F2 (0.40) ALDH1A1
SCHEMBL6236337 0.78 MEN1 (0.55) KIF11MEN1KMT2ALMNAHTT
SCHEMBL9494550 0.78 TDP1 (0.43) ALDH1A1CA12CA1
SCHEMBL2255790 0.77 ALDH1A1 (0.64) ALDH1A1MEN1KMT2ALMNAHTT
SCHEMBL21542302 0.76 MEN1 (0.54) KIF11MEN1KMT2ALMNAHTT
SCHEMBL11941008 0.76 HDAC1 (0.39) KIF11ALDH1A1MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2212277-A1 AMINE LINKED MODULATORS OF Y-SECRETASE Janssen Pharmaceutica, N.V. (BE) 2010-08-04 EP disclosed
WO-2009052350-A1 AMINE LINKED MODULATORS OF Y-SECRETASE JANSSEN PHARMACEUTICA, N.V. (BE) 2009-04-23 WO disclosed