SCHEMBL365595

SCHEMBL365595

O=C(Nc1ccc(Oc2ccc(F)cc2)cc1)c1ccccn1

nearest known ligand 0.77

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.68
RAB9A P51151 3/20 0.68
SMN1; SMN2 Q16637 3/20 0.68
PKM P14618 2/20 0.68
MAPT P10636 2/20 0.68
KDM4E B2RXH2 1/20 0.64
MITF O75030 1/20 0.64
KDR P35968 1/20 0.62
KMT2A Q03164 1/20 0.61
GRM4 Q14833 7/20 0.56
GAA P10253 1/20 0.56
AXL P30530 1/20 0.55
PTGS1 P23219 1/20 0.53
PTGS2 P35354 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30686047 0.91 GRM4 (0.65) NPC1RAB9ASMN1; SMN2PKMMAPT
SCHEMBL10415452 0.91 GRM4 (0.65) NPC1RAB9ASMN1; SMN2PKMMAPT
SCHEMBL2535716 0.85 GRM4 (0.67) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL3092361 0.81 SMN1; SMN2 (1.00) NPC1RAB9ASMN1; SMN2PKMMAPT
SCHEMBL2533682 0.80 NPC1 (0.71) NPC1RAB9ASMN1; SMN2PKMMAPT
SCHEMBL30904871 0.80 NPC1 (0.71) NPC1RAB9ASMN1; SMN2PKMMAPT
SCHEMBL27930549 0.79 PTGS1 (0.56) NPC1RAB9ASMN1; SMN2PKMMAPT
SCHEMBL6630361 0.78 NPC1 (0.69) NPC1RAB9ASMN1; SMN2PKMMAPT
SCHEMBL8215155 0.78 NPC1 (0.51) NPC1RAB9ASMN1; SMN2PKMMAPT
SCHEMBL231897 0.78 KDR (0.78) NPC1RAB9ASMN1; SMN2PKMMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593434-A1 PYRIDINE COMPOUNDS AS SODIUM CHANNEL BLOCKERS Purdue Pharma LP (US) 2013-05-22 EP disclosed
WO-2012007836-A1 PYRIDINE COMPOUNDS AS SODIUM CHANNEL BLOCKERS PURDUE PHARMA .LP. (US) 2012-01-19 WO disclosed