SCHEMBL3657153

SCHEMBL3657153

C[C@H](CC#CC(N)CCF)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.46
GRM5 P41594 1/20 0.41
AOC3 Q16853 2/20 0.39
RIPK1 Q13546 1/20 0.38
HTR2A P28223 1/20 0.37
TRPA1 O75762 2/20 0.36
SLC7A5 Q01650 1/20 0.35
HRH1 P35367 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6063975 0.80 TAAR1 (0.50) TAAR1GRM5AOC3RIPK1HTR2A
SCHEMBL6014502 0.74 TAAR1 (0.57) TAAR1GRM5AOC3RIPK1HTR2A
SCHEMBL3627864 0.73 TAAR1 (0.60) TAAR1AOC3RIPK1TRPA1HRH1
SCHEMBL6014574 0.72 TAAR1 (0.54) TAAR1GRM5AOC3RIPK1HTR2A
SCHEMBL2480450 0.70 TAAR1 (0.47) TAAR1
SCHEMBL18244887 0.69 GRM5 (0.50) TAAR1GRM5AOC3RIPK1HTR2A
SCHEMBL19374761 0.66 TAAR1 (0.56) TAAR1AOC3RIPK1HTR2ATRPA1
SCHEMBL23336071 0.66 TAAR1 (0.67) TAAR1AOC3RIPK1HTR2ATRPA1
SCHEMBL1281 0.66 TAAR1 (0.67) TAAR1AOC3RIPK1HTR2ATRPA1
SCHEMBL5791734 0.66 TAAR1 (0.67) TAAR1AOC3RIPK1HTR2ATRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2217549-A2 COMPOUNDS FOR USE IN IMAGING, DIAGNOSING, AND/OR TREATMENT OF DISEASES OF THE CENTRAL NERVOUS SYSTEM OR OF TUMORS Bayer Schering Pharma Aktiengesellschaft (DE) 2010-08-18 EP disclosed
WO-2009052970-A2 COMPOUNDS FOR USE IN IMAGING, DIAGNOSING, AND/OR TREATMENT OF DISEASES OF THE CENTRAL NERVOUS SYSTEM OR OF TUMORS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-04-30 WO disclosed