SCHEMBL3659404

SCHEMBL3659404

Cc1ccc(-c2cc(C(=O)NC[C@H](C)O)cc(-c3ccnn3CC3CC3)c2)nc1

nearest known ligand 0.43

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 15/20 0.43
P2RX2 Q9UBL9 15/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14837447 0.88 P2RX3 (0.45) P2RX3P2RX2
SCHEMBL27846532 0.86 P2RX3 (0.56) P2RX3P2RX2
SCHEMBL3659401 0.86 P2RX3 (0.56) P2RX3P2RX2
SCHEMBL3664334 0.86 P2RX3 (0.52) P2RX3P2RX2
SCHEMBL3660665 0.85 P2RX3 (0.59) P2RX3P2RX2
SCHEMBL3658272 0.84 P2RY14 (0.38) P2RX3P2RX2
SCHEMBL3663110 0.84 P2RX3 (0.39) P2RX3P2RX2
SCHEMBL3660372 0.84 P2RX3 (0.45) P2RX3P2RX2
SCHEMBL4163451 0.83 P2RX3 (0.58) P2RX3P2RX2
SCHEMBL3660190 0.83 P2RX3 (0.60) P2RX3P2RX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234976-A1 NOVEL PYRAZOLE-SUBSTITUTED ARYLAMIDES F. Hoffmann-La Roche AG (CH) 2010-10-06 EP disclosed
WO-2009077367-A1 NOVEL PYRAZOLE-SUBSTITUTED ARYLAMIDES F. HOFFMANN-LA ROCHE AG (CH) 2009-06-25 WO disclosed