SCHEMBL365987

SCHEMBL365987

[C]1=CC2Nc3ccccc3C=CC2C=C1

nearest known ligand 0.34

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL367177 0.87 GAA (0.34) GAAMAPT
SCHEMBL3118101 0.76 GAA (0.39) GAAMAPT
SCHEMBL11993899 0.69 GAA (0.35) GAAMAPT
SCHEMBL5737091 0.65
SCHEMBL4445110 0.65 GAA (0.34) GAAMAPT
SCHEMBL367620 0.65 GAA (0.34) GAAMAPT
SCHEMBL17602387 0.65 IDO1 (0.43)
SCHEMBL4540870 0.64 GAA (0.44) GAAMAPT
SCHEMBL12159337 0.64 GAA (0.44) GAAMAPT
SCHEMBL6056252 0.64 GAA (0.44) GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 62 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4392168-A1 IONIC LIQUID-BASED COMPOSITE MEMBRANES USING FUNCTIONAL CROSS-LINKERS The Regents of the University of Colorado, a body corporate (US) 2024-07-03 EP disclosed
WO-2024081715-A2 LIPID NANOPARTICLE (LNP) COMPOSITIONS FOR PLACENTA-SELECTIVE CARGO DELIVERY, AND METHODS OF USE THEREOF THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2024-04-18 WO disclosed
WO-2023028323-A9 IONIC LIQUID-BASED COMPOSITE MEMBRANES USING FUNCTIONAL CROSS-LINKERS THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2024-04-04 WO disclosed
WO-2023240081-A1 TREATMENT, AMELIORATION, AND/OR PREVENTION OF INFLAMMATORY AND AUTOIMMUNE DISEASES YALE UNIVERSITY (US) 2023-12-14 WO disclosed
EP-4216949-A1 SELECTIVE AGONISTS OF 5-HT2A RECEPTOR AND METHODS OF USE Yale University (US) 2023-08-02 EP disclosed
WO-2023056282-A1 COMPOSITIONS AND METHODS FOR T CELL TARGETED DELIVERY OF THERAPEUTIC AGENTS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2023-04-06 WO disclosed
WO-2023049806-A1 COMPOUNDS AND METHODS FOR TREATING CANCERS THAT ARE MGMT DEFICIENT REGARDLESS OF MMR STATUS YALE UNIVERSITY (US) 2023-03-30 WO disclosed
WO-2023028323-A1 IONIC LIQUID-BASED COMPOSITE MEMBRANES USING FUNCTIONAL CROSS-LINKERS THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2023-03-02 WO disclosed
WO-2022150584-A1 NON-COVALENT INHIBITORS OF THE MAIN PROTEASE OF SARS-COV-2 AND METHODS OF USE YALE UNIVERSITY (US) 2022-07-14 WO disclosed
WO-2020257753-A1 PHOSPHATIDYLSERINE DECARBOXYLASE INHIBITORS YALE UNIVERSITY (US) 2020-12-24 WO disclosed
EP-2134689-A2 INHIBITORS OF FOCAL ADHESION KINASE The Scripps Research Institute (US) 2009-12-23 EP disclosed
WO-2009139834-A1 BIOACTIVE COMPOUNDS FOR TREATMENT OF CANCER AND NEURODEGENERATIVE DISEASES PONIARD PHARMACEUTICALS, INC. (US) 2009-11-19 WO disclosed
WO-2009102876-A1 MACROCYCLIC INHIBITORS OF HEPATITIS C PROTEASE PHENOMIX CORPORATION (US) 2009-08-20 WO disclosed
WO-2009079008-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS FENG YANGBO (US) 2009-06-25 WO disclosed
WO-2009079009-A1 ANILIDES AND ANALOGS AS RHO KINASE INHIBITORS FENG YANGBO (US) 2009-06-25 WO disclosed
WO-2009079011-A1 BENZIMIDAZOLES AND ANALOGS AS RHO KINASE INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 2009-06-25 WO disclosed
WO-2008115369-A2 INHIBITORS OF FOCAL ADHESION KINASE THE SCRIPPS RESEARCH INSTITUTE (US) 2008-09-25 WO disclosed
EP-1689757-A4 HETEROCYCLIC BORONIC ACID COMPOUNDS PHENOMIX CORP (US) 2007-01-10 EP disclosed
EP-1689757-A1 HETEROCYCLIC BORONIC ACID COMPOUNDS Phenomix Corporation (US) 2006-08-16 EP disclosed
WO-2005047297-A1 HETEROCYCLIC BORONIC ACID COMPOUNDS PHENOMIX CORPORATION (US) 2005-05-26 WO disclosed