SCHEMBL3660948

SCHEMBL3660948

CCCc1nc(-c2nccs2)cc(C(N)=O)c1Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE11A Q9HCR9 1/20 0.43
TACR3 P29371 1/20 0.39
HPGD P15428 11/20 0.39
MCL1 Q07820 1/20 0.36
ADORA2A P29274 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3660945 0.93 PDE11A (0.44) PDE11ATACR3HPGDMCL1ADORA2A
SCHEMBL3347230 0.71 CHEK2 (0.41) HPGDHDAC3HDAC4HDAC1HDAC6
SCHEMBL28139104 0.70 PDPK1 (0.40) NPC1RAB9A
SCHEMBL28843050 0.70 PLA2G2A (0.44) NPC1RAB9A
SCHEMBL3350744 0.68 HPGD (0.37) HPGDNPC1RAB9AMEN1KMT2A
Hydrochloric Acid SCHEMBL3349083 0.67 HPGD (0.36) HPGDNPC1RAB9AMEN1KMT2A
Hydrochloric Acid SCHEMBL3351578 0.67 HPGD (0.36) HPGDNPC1RAB9AMEN1KMT2A
SCHEMBL13957931 0.64 TACR3 (0.62) TACR3HPGDNPC1RAB9AMEN1
SCHEMBL13729456 0.64 PDPK1 (0.40) HDAC3HDAC4HDAC1HDAC6
SCHEMBL28255768 0.64 FFAR1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7838676-B2 Beta-secretase modulators and methods of use AMGEN INC. (US) 2010-11-23 US disclosed