SCHEMBL3661014

SCHEMBL3661014

CC(=O)NC(C)(C)c1cc(-c2cncc(Br)c2)cc(-c2ccccn2)n1.CCN(C)c1cc(-c2cncc(Br)c2)cc(-c2ccccn2)n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.33
RXFP1 Q9HBX9 2/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 3/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
PTPN7 P35236 1/20 0.33
DUSP3 P51452 1/20 0.33
HDAC1 Q13547 3/20 0.32
GPR39 O43194 2/20 0.32
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
ESR1 P03372 1/20 0.31
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
KMT2A Q03164 2/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3664633 0.90 NPSR1 (0.37) NPSR1RXFP1ALDH1A1LMNAKDM4E
SCHEMBL3665505 0.85 ESR1 (0.37) NPSR1RXFP1ALDH1A1LMNAPTPN7
SCHEMBL3663869 0.76 GRM5 (0.36) NPSR1RXFP1ALDH1A1LMNAKDM4E
SCHEMBL3664991 0.76 MDM2 (0.41) NPSR1RXFP1ALDH1A1LMNAMAPT
SCHEMBL4183866 0.74 CYP2A6 (0.36) NPSR1RXFP1ALDH1A1LMNAKDM4E
SCHEMBL3667875 0.69 GPR39 (0.37) NPSR1RXFP1ALDH1A1LMNAKDM4E
SCHEMBL3663765 0.66 CCR1 (0.40) NPSR1RXFP1ALDH1A1LMNAKDM4E
SCHEMBL3663615 0.65 CCR1 (0.37) NPSR1RXFP1ALDH1A1LMNAKDM4E
SCHEMBL3661769 0.65 KDM4E (0.37) NPSR1RXFP1ALDH1A1LMNAKDM4E
SCHEMBL3659080 0.65 CYP1A2 (0.45) NPSR1RXFP1ALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2242742-A2 ORGANIC COMPOUNDS Novartis AG (CH) 2010-10-27 EP disclosed
WO-2009087212-A2 PYRIDINE DERIVATIVES NOVARTIS AG (CH) 2009-07-16 WO disclosed