SCHEMBL3661174

SCHEMBL3661174

CCOC(=O)CC1CCCc2cnc(Nc3ccc(-c4nc(C)c[nH]4)c(OC)c3)nc21

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 9/20 0.37
BRD4 O60885 1/20 0.36
PAK1 Q13153 1/20 0.36
PTK2 Q05397 1/20 0.35
FYN P06241 1/20 0.35
CDK2 P24941 2/20 0.35
CDK9 P50750 2/20 0.35
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
IKBKB O14920 1/20 0.34
TTK P33981 1/20 0.34
KDR P35968 2/20 0.34
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34
PDGFRB P09619 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3664695 0.88 PLK1 (0.39) PLK1BRD4PAK1PTK2FYN
SCHEMBL3660797 0.84 PLK1 (0.38) PLK1FYNCDK2KDRPSEN1
SCHEMBL3657821 0.84 PLK1 (0.39) PLK1PTK2CDK2KDRPSEN1
SCHEMBL3665907 0.82 PLK1 (0.39) PLK1PTK2CDK2KDRPSEN1
SCHEMBL1616552 0.82 PSEN1 (0.52) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3662116 0.82 PDGFRB (0.39) PLK1BRD4FYNKDRPSEN1
SCHEMBL3661161 0.81 PLK1 (0.38) PLK1CDK2KDRPSEN1PSEN2
SCHEMBL3665261 0.80 PLK1 (0.38) PLK1CDK2KDRPSEN1PSEN2
SCHEMBL3659836 0.80 PLK1 (0.38) PLK1CDK2CDK9IKBKBKDR
SCHEMBL3664634 0.80 PSEN1 (0.39) PLK1BRD4PTK2CDK2PSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2231629-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-09-29 EP disclosed
WO-2009087127-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-07-16 WO disclosed