SCHEMBL3661558

SCHEMBL3661558

Cc1ccc(-c2oncc2C(=O)N2CCC[C@H](C(C)(C)O)C2I)cc1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 14/20 0.39
HCRTR1 O43613 12/20 0.39
SLC22A12 Q96S37 1/20 0.35
GRM5 P41594 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3665234 1.00 HCRTR2 (0.39) HCRTR2HCRTR1SLC22A12GRM5ALDH1A1
SCHEMBL3656862 0.91 GRM5 (0.42) HCRTR2HCRTR1SLC22A12GRM5ALDH1A1
SCHEMBL3658400 0.91 GRM5 (0.42) HCRTR2HCRTR1SLC22A12GRM5ALDH1A1
SCHEMBL3663269 0.91 TRPV1 (0.36) HCRTR2HCRTR1GRM5LMNASMN1; SMN2
SCHEMBL3665267 0.91 TRPV1 (0.36) HCRTR2HCRTR1GRM5LMNASMN1; SMN2
SCHEMBL3664407 0.89 HCRTR2 (0.41) HCRTR2HCRTR1GRM5
SCHEMBL3666816 0.89 HCRTR2 (0.41) HCRTR2HCRTR1GRM5
SCHEMBL3661305 0.86 HCRTR2 (0.41) HCRTR2HCRTR1
SCHEMBL3663469 0.86 HCRTR2 (0.41) HCRTR2HCRTR1
SCHEMBL3663295 0.84 HCRTR1 (0.39) HCRTR2HCRTR1LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2231650-A1 ISOXAZOLE DERIVATIVES AS MODULATORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 Biovitrum AB (publ) (SE) 2010-09-29 EP disclosed
WO-2009090239-A1 ISOXAZOLE DERIVATIVES AS MODULATORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (PUBL) (SE) 2009-07-23 WO disclosed