SCHEMBL3662458

SCHEMBL3662458

COc1cccc(OC)c1C(=O)N(C(=O)OC(C)(C)C)C1CCNC1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 14/20 0.42
SLC6A2 P23975 12/20 0.42
SLC6A3 Q01959 10/20 0.42
CYP2D6 P10635 7/20 0.42
KCNH2 Q12809 6/20 0.42
MBTPS1 Q14703 5/20 0.41
F10 P00742 1/20 0.41
PLAU P00749 1/20 0.41
REN P00797 1/20 0.40
CHRM3 P20309 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1868079 0.75 SLC6A4 (0.38) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL5506061 0.75 SLC6A4 (0.38) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL1868080 0.75 SLC6A4 (0.38) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL5506058 0.75 SLC6A4 (0.38) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL6526760 0.73 SLC6A4 (0.37) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL28482383 0.73 MEN1 (0.42) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL20791408 0.71 SLC6A4 (0.57) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL17868819 0.70 SLC6A2 (0.57) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL5823064 0.69 TACR1 (0.48) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL16964830 0.69 SLC6A4 (0.43) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234999-A1 HETEROARYL DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2010-10-06 EP disclosed
WO-2009080533-A1 HETEROARYL DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-07-02 WO disclosed