SCHEMBL366289

SCHEMBL366289

O=C(O)c1ccc(Cc2ccc(Cl)c(Cl)c2)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HAO1 Q9UJM8 1/20 0.67
TSHR P16473 2/20 0.62
EPHX2 P34913 1/20 0.59
SRD5A2 P31213 4/20 0.59
RXRA P19793 1/20 0.50
RXRB P28702 1/20 0.50
RXRG P48443 1/20 0.50
SLC6A2 P23975 2/20 0.49
SLC6A4 P31645 2/20 0.49
SLC6A3 Q01959 2/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
HPGD P15428 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
ALDH1A1 P00352 2/20 0.47
ALOX15 P16050 1/20 0.47
RNASEH1 O60930 1/20 0.47
TBXA2R P21731 1/20 0.47
PTGER1 P34995 1/20 0.47
PTGER4 P35408 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11224189 0.84 KMT2A (0.68) HAO1TSHREPHX2SLC6A2SLC6A4
SCHEMBL68390 0.82 SRD5A2 (0.69) TSHRSRD5A2RXRARXRBRXRG
SCHEMBL16363560 0.81 HAO1 (0.58) HAO1TSHREPHX2SLC6A2SLC6A4
SCHEMBL11361475 0.81 HAO1 (0.58) HAO1TSHRSLC6A2SLC6A4SLC6A3
SCHEMBL27873324 0.80 TSHR (0.56) HAO1TSHREPHX2SRD5A2SLC6A2
SCHEMBL11221375 0.80 HAO1 (1.00) HAO1TSHREPHX2SLC6A2SLC6A4
SCHEMBL11467697 0.80 TSHR (0.74) TSHRSRD5A2ALDH1A1ALOX15MEN1
SCHEMBL11673315 0.80 SRD5A2 (0.62) TSHRSRD5A2RXRARXRBRXRG
Hydrochloric Acid SCHEMBL25188150 0.80 SRD5A2 (0.67) TSHRSRD5A2RXRARXRBRXRG
Hydrochloric Acid SCHEMBL7133360 0.80 SRD5A2 (0.67) TSHRSRD5A2RXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593427-B1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LTD (GB) 2014-12-24 EP disclosed
EP-2593427-A1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN Pfizer Limited (GB) 2013-05-22 EP disclosed
WO-2012007883-A1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LIMITED (GB) 2012-01-19 WO disclosed
WO-2012007883-A1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LIMITED (GB) 2012-01-19 WO disclosed
US-20120010207-A1 Chemical Compounds PFIZER LIMITED (GB) 2012-01-12 US disclosed
US-20120010207-A1 Chemical Compounds PFIZER LIMITED (GB) 2012-01-12 US disclosed
US-20120010207-A1 Chemical Compounds PFIZER LIMITED (GB) 2012-01-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120010207-A1 Chemical Compounds SCN1A, SCN1B, SCN7A HAO1 2919/4885TSHR 2473/4885EPHX2 3890/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.