SCHEMBL3663522

SCHEMBL3663522

N#Cc1ccccc1-c1nc(COc2ccc3c(=O)c(-c4ccc(O)cc4)coc3c2)no1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ALDH2 P05091 19/20 0.55
MAOA P21397 10/20 0.55
MAOB P27338 10/20 0.55
XDH P47989 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2108020 0.87 ALDH2 (0.61) ALDH2MAOAMAOB
SCHEMBL3666659 0.86 ALDH2 (0.59) ALDH2MAOAMAOB
SCHEMBL2106711 0.86 ALDH2 (0.54) ALDH2MAOAMAOBXDH
SCHEMBL2107604 0.86 XDH (0.57) ALDH2MAOAMAOBXDH
SCHEMBL2106733 0.84 ALDH2 (0.57) ALDH2MAOAMAOBXDH
SCHEMBL2108143 0.83 ALDH2 (0.60) ALDH2MAOAMAOBXDH
SCHEMBL4090316 0.83 XDH (0.66) ALDH2MAOAMAOBXDH
SCHEMBL3631565 0.82 ALDH2 (0.65) ALDH2MAOAMAOBXDH
SCHEMBL2108533 0.81 ALDH2 (0.59) ALDH2MAOAMAOB
SCHEMBL2107605 0.81 ALDH2 (0.56) ALDH2MAOAMAOBXDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2254878-A1 ALDH-2 INHIBITORS IN THE TREATMENT OF ADDICTION Gilead Palo Alto, Inc. (US) 2010-12-01 EP disclosed
EP-2231149-A2 ALDH-2 INHIBITORS IN THE TREATMENT OF PSYCHIATRIC DISORDERS CV Therapeutics Inc. (US) 2010-09-29 EP disclosed
WO-2009094028-A1 ALDH-2 INHIBITORS IN THE TREATMENT OF ADDICTION CV THERAPEUTICS, INC. (US) 2009-07-30 WO disclosed
WO-2009061924-A2 ALDH-2 INHIBITORS IN THE TREATMENT OF PSYCHIATRIC DISORDERS CV THERAPEUTICS, INC. (US) 2009-05-14 WO disclosed
EP-2046769-A2 ALDH-2 INHIBITORS IN THE TREATMENT OF ADDICTION CV THERAPEUTICS, INC. (US) 2009-04-15 EP disclosed
WO-2008014497-A2 ALDH-2 INHIBITORS IN THE TREATMENT OF ADDICTION CV THERAPEUTICS, INC. (US) 2008-01-31 WO disclosed