SCHEMBL3663531

SCHEMBL3663531

CC(C)(C)OC(=O)NCCCCCCCCCCCCN(C(N)=NC#N)c1ccncc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
CYP3A4 P08684 1/20 0.41
CSNK2A2 P19784 1/20 0.40
CSNK2A1 P68400 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CA1 P00915 7/20 0.39
CA2 P00918 7/20 0.39
CA12 O43570 5/20 0.39
CA9 Q16790 5/20 0.39
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
MAPT P10636 1/20 0.37
RAB9A P51151 1/20 0.37
LATS1 O95835 1/20 0.36
BRD4 O60885 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
DRD2 P14416 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6955341 0.83 MAOA (0.46) MAOAMAOBCYP3A4CSNK2A2CSNK2A1
SCHEMBL6953013 0.83 MAOA (0.46) MAOAMAOBCYP3A4CSNK2A2CSNK2A1
SCHEMBL809997 0.80 PLG (0.33)
SCHEMBL810674 0.80 PLG (0.33)
SCHEMBL17074729 0.77 CA12 (0.33) MAOAMAOBTDP1CA1CA2
SCHEMBL6949199 0.76 IKBKB (0.46) MAOAMAOBCYP3A4CSNK2A2CSNK2A1
SCHEMBL810259 0.76 IKBKB (0.46) MAOAMAOBCYP3A4CSNK2A2CSNK2A1
Hydrochloric Acid SCHEMBL3666361 0.76 MAOA (0.32) MAOAMAOBCA1CA2CA12
SCHEMBL7070178 0.74 CYP3A4 (0.44) MAOAMAOBCYP3A4CSNK2A2CSNK2A1
SCHEMBL4420719 0.70 CYP3A4 (0.44) CYP3A4CSNK2A2CSNK2A1TDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197443-A2 COMPOSITIONS AND METHODS FOR EFFECTING NAD+ LEVELS USING A NICOTINAMIDE PHOSPHORIBOSYL TRANSFERASE INHIBITOR Gemin X Pharmaceuticals Canada Inc. (CA) 2010-06-23 EP claimed
WO-2009072004-A2 COMPOSITIONS AND METHODS FOR EFFECTING NAD+ LEVELS USING A NICOTINAMIDE PHOSPHORIBOSYL TRANSFERASE INHIBITOR GEMIN X PHARMACEUTICALS CANADA, INC. (US) 2009-06-11 WO claimed
EP-2197443-A2 COMPOSITIONS AND METHODS FOR EFFECTING NAD+ LEVELS USING A NICOTINAMIDE PHOSPHORIBOSYL TRANSFERASE INHIBITOR Gemin X Pharmaceuticals Canada Inc. (CA) 2010-06-23 EP disclosed
WO-2009072004-A2 COMPOSITIONS AND METHODS FOR EFFECTING NAD+ LEVELS USING A NICOTINAMIDE PHOSPHORIBOSYL TRANSFERASE INHIBITOR GEMIN X PHARMACEUTICALS CANADA, INC. (US) 2009-06-11 WO disclosed