SCHEMBL3663651

SCHEMBL3663651

CC(c1ccccc1)c1ccccc1C(N)=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.47
ALOX5 P09917 1/20 0.44
PARP1 P09874 1/20 0.44
BCAT2 O15382 1/20 0.44
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 2/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
HSD17B10 Q99714 1/20 0.44
TYR P14679 1/20 0.43
GAA P10253 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
SRC P12931 1/20 0.42
AURKA O14965 2/20 0.42
RPS6KB1 P23443 2/20 0.42
NOS2 P35228 1/20 0.42
AURKB Q96GD4 1/20 0.42
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5968855 1.00 IRAK4 (0.47) IRAK4ALOX5PARP1BCAT2ALDH1A1
SCHEMBL6266294 1.00 IRAK4 (0.47) IRAK4ALOX5PARP1BCAT2ALDH1A1
SCHEMBL9783644 0.88 IRAK4 (0.53) IRAK4PARP1BCAT2ALDH1A1KDM4E
SCHEMBL27971185 0.88 ALDH1A1 (0.48) IRAK4ALOX5PARP1ALDH1A1KDM4E
SCHEMBL27971183 0.88 ALDH1A1 (0.48) IRAK4ALOX5PARP1ALDH1A1KDM4E
SCHEMBL27971184 0.88 ALDH1A1 (0.48) IRAK4ALOX5PARP1ALDH1A1KDM4E
SCHEMBL584940 0.86 ALDH1A1 (0.55) ALDH1A1KDM4EMAPTHPGDHSD17B10
SCHEMBL21835618 0.86 IRAK4 (0.42) IRAK4ALOX5PARP1BCAT2ALDH1A1
SCHEMBL27511285 0.86 IRAK4 (0.42) IRAK4ALOX5PARP1BCAT2ALDH1A1
SCHEMBL20425250 0.86 IRAK4 (0.42) IRAK4ALOX5PARP1BCAT2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3724325-A1 CARBOXYESTERASE POLYPEPTIDES FOR AMIDE COUPLING Codexis, Inc. (US) 2020-10-21 EP claimed
WO-2019118557-A1 CARBOXYESTERASE POLYPEPTIDES FOR AMIDE COUPLING CODEXIS, INC. (US) 2019-06-20 WO claimed
WO-2023018473-A1 COMBINED DETERMINATION OF THE CONCENTRATION AND ENANTIOMERIC COMPOSITION OF CHIRAL COMPOUNDS USING SINGLE CHIROPTICAL ASSAY GEORGETOWN UNIVERSITY (US) 2023-02-16 WO disclosed
CN-102964195-B Method for preparing second-level and third-level substituted amide UNIV WENZHOU 2015-06-24 CN disclosed
CN-102964195-A Method for preparing second-level and third-level substituted amide UNIV WENZHOU 2013-03-13 CN disclosed
EP-2234995-A1 LEUKOTRIENE B4 INHIBITORS F. Hoffmann-La Roche AG (CH) 2010-10-06 EP disclosed
WO-2009077385-A1 LEUKOTRIENE B4 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2009-06-25 WO disclosed
EP-1960350-A1 NEW N-(1-METHYL-2PHENYLETHYL)BENZAMIDE DERIVATIVES BAYER CROPSCIENCE SA (FR) 2008-08-27 EP disclosed
WO-2007060162-A1 NEW N-(1-METHYL-2PHENYLETHYL)BENZAMIDE DERIVATIVES BAYER CROPSCIENCE SA (FR) 2007-05-31 WO disclosed
EP-1509499-A1 PYRROLE COMPOUNDS FOR THE TREATMENT OF PROSTAGLANDIN MEDIATED DISEASES GLAXO GROUP LIMITED (GB) 2005-03-02 EP disclosed
WO-2003101959-A1 PYRROLE COMPOUNDS FOR THE TREATMENT OF PROSTAGLANDIN MEDIATED DISEASES GLAXO GROUP LIMITED (GB) 2003-12-11 WO disclosed
EP-0078845-A4 ANTI-CONVULSANT. CLARK CHARLES RANDALL 1983-09-02 EP disclosed
EP-0078845-A1 ANTI-CONVULSANT. CLARK CHARLES RANDALL 1983-05-18 EP disclosed
WO-1982004046-A1 ANTI-CONVULSANT CLARK CHARLES RANDALL 1982-11-25 WO disclosed