SCHEMBL3664375

SCHEMBL3664375

C=C(c1ccccc1)c1ccc2[nH]c3ncc(Cl)cc3c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2 P11137 1/20 0.43
JAK2 O60674 1/20 0.41
CCKBR P32239 1/20 0.39
CHEK1 O14757 2/20 0.38
KDR P35968 1/20 0.38
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38
ERBB2 P04626 1/20 0.35
PTK6 Q13882 1/20 0.35
CSF1R P07333 1/20 0.35
GABRP O00591 2/20 0.35
GABRD O14764 2/20 0.35
GABRA1 P14867 2/20 0.35
GABRB1 P18505 2/20 0.35
GABRG2 P18507 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL676282 0.85 MAPT (0.45) KDRGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL674851 0.84 MAP2 (0.49) MAP2JAK2CCKBRGRIN2DGRIN3B
SCHEMBL674860 0.84 SMN1; SMN2 (0.38) MAP2JAK2CCKBRGRIN2DGRIN3B
SCHEMBL674892 0.81 KDM4E (0.48) MAP2CCKBRERBB2PTK6GABRP
SCHEMBL675814 0.81 GABRP (0.44) CCKBRGABRPGABRDGABRA1GABRB1
SCHEMBL11860308 0.80 KDR (0.46) CHEK1KDRKMT2AMEN1RAB9A
SCHEMBL676824 0.79 KDM4E (0.42) CCKBRCHEK1KDRGRIN2DGRIN3B
SCHEMBL3669225 0.78 AURKA (0.47) CHEK1KDRERBB2PTK6
SCHEMBL675229 0.77 ERBB2 (0.53) MAP2CCKBRCHEK1ERBB2PTK6
SCHEMBL15873503 0.76 CHUK (0.54) MAP2JAK2CHEK1KDRCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2161271-A1 Alpha-carboline inhibitors of NMP-ALK, RET, and Bcr-Abl Università Degli Studi Di Milano - Bicocca (IT) 2010-03-10 EP disclosed