SCHEMBL3664848

SCHEMBL3664848

COc1ccccc1C1CCCC(Br)C1=O.COc1ccccc1C1CCCCC1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.39
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
USP2 O75604 1/20 0.39
TNKS O95271 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38
HTR2C P28335 2/20 0.37
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
ALDH1A1 P00352 3/20 0.36
MAPT P10636 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
PKM P14618 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
POLL Q9UGP5 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
RECQL P46063 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1616195 0.91 MEN1 (0.45) CYP19A1MEN1KMT2AUSP2HTR2C
SCHEMBL15874851 0.88 CYP19A1 (0.47) CYP19A1MEN1KMT2AUSP2TNKS
SCHEMBL1616886 0.88 CYP19A1 (0.47) CYP19A1MEN1KMT2AUSP2TNKS
SCHEMBL30496207 0.88 CYP19A1 (0.47) CYP19A1MEN1KMT2AUSP2TNKS
SCHEMBL512007 0.84 CYP19A1 (0.48) CYP19A1MEN1KMT2AUSP2HTR2C
SCHEMBL3662535 0.73 MAOA (0.33) MEN1KMT2AUSP2ALDH1A1
SCHEMBL19993899 0.72 HCRTR1 (0.40) MEN1KMT2AUSP2HCRTR1HCRTR2
SCHEMBL17185892 0.70 TP53 (0.43) HTR2CCA1CA2CA4CA6
SCHEMBL4918535 0.69 TP53 (0.46) MEN1KMT2AALDH1A1MAPTTDP1
SCHEMBL1616342 0.69 TP53 (0.41) HTR2CALDH1A1CA1CA2RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2231629-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-09-29 EP disclosed
WO-2009087127-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-07-16 WO disclosed