SCHEMBL3665609

SCHEMBL3665609

CS(=O)(=O)OC1CCN(c2nc3ccc(-c4ccc(C#N)cc4)cc3s2)C1I

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.41
NR1H3 Q13133 1/20 0.41
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HRH3 Q9Y5N1 3/20 0.38
KCNH2 Q12809 1/20 0.36
CA12 O43570 3/20 0.35
CA2 P00918 3/20 0.35
CA9 Q16790 3/20 0.35
PIK3CG P48736 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CTSK P43235 1/20 0.34
USP30 Q70CQ3 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1095382 0.80 HRH3 (0.44) NR1H2NR1H3MAPTKMT2ANPSR1
SCHEMBL1095813 0.80 HRH3 (0.44) NR1H2NR1H3MAPTKMT2ANPSR1
SCHEMBL1095383 0.80 HRH3 (0.44) NR1H2NR1H3MAPTKMT2ANPSR1
SCHEMBL3665269 0.76 RAB9A (0.47) NR1H2NR1H3MAPTNPC1RAB9A
SCHEMBL1094234 0.68 HRH3 (0.50) MAPTKMT2ANPSR1HRH3KCNH2
SCHEMBL1096234 0.68 HRH3 (0.50) MAPTKMT2ANPSR1HRH3KCNH2
SCHEMBL1094232 0.68 HRH3 (0.50) MAPTKMT2ANPSR1HRH3KCNH2
SCHEMBL1094449 0.67 HRH3 (0.45) NR1H2NR1H3MAPTKMT2ANPSR1
SCHEMBL1094450 0.67 HRH3 (0.45) NR1H2NR1H3MAPTKMT2ANPSR1
SCHEMBL1095586 0.66 HRH3 (0.65) HRH3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2237779-A1 BENZOTHIAZOLE AND BENZOXAZOLE DERIVATIVES AND METHODS OF USE Abbott Laboratories (US) 2010-10-13 EP disclosed
WO-2009085945-A1 BENZOTHIAZOLE AND BENZOXAZOLE DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2009-07-09 WO disclosed