SCHEMBL367128

SCHEMBL367128

CC(OC(=O)c1c2ccccc2n2cc(OCC#N)ccc12)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.35
TP53 P04637 1/20 0.35
HSD17B10 Q99714 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
GABRA4 P48169 1/20 0.35
GABRA6 Q16445 1/20 0.35
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
PPARG P37231 1/20 0.34
SRD5A1 P18405 3/20 0.34
SRD5A2 P31213 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364154 0.90 MAPT (0.39) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL366259 0.88 ALDH1A1 (0.36) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL366083 0.87 PSEN1 (0.38) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL365124 0.86 FLT3 (0.35) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL367500 0.86 PSEN1 (0.35) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL366403 0.86 KDM4E (0.37) ALDH1A1HSD17B10PSEN1PSEN2APH1B
SCHEMBL367591 0.85 PSEN1 (0.35) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL366563 0.85 TSHR (0.40) ALDH1A1HSD17B10PSEN1PSEN2APH1B
SCHEMBL367127 0.84 ALDH1A1 (0.48) ALDH1A1TP53HSD17B10GABRA1GABRG2
SCHEMBL364973 0.84 KMT2A (0.42) ALDH1A1PSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed