SCHEMBL3673050

SCHEMBL3673050

Cc1c(Cl)cccc1C(c1ccccn1)c1cnc[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 10/20 0.46
ADRA2B P18089 10/20 0.46
ADRA2C P18825 10/20 0.46
ADRA1A P35348 7/20 0.46
ADRA1B P35368 6/20 0.46
ADRA1D P25100 5/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2D6 P10635 2/20 0.46
KCNH2 Q12809 1/20 0.46
TP53 P04637 1/20 0.46
CYP2C9 P11712 1/20 0.46
TSHR P16473 1/20 0.46
CYP2C19 P33261 1/20 0.46
SLC6A2 P23975 1/20 0.45
HTR7 P34969 1/20 0.45
HRH3 Q9Y5N1 2/20 0.42
HRH4 Q9H3N8 1/20 0.42
MEN1 O00255 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3061266 0.87 ADRA2A (0.41) ADRA2AADRA2BADRA2CADRA1AADRA1B
SCHEMBL3067675 0.85 HRH3 (0.42) ADRA2AADRA2BADRA2CADRA1AADRA1B
SCHEMBL3051753 0.85 ADRA2A (0.46) ADRA2AADRA2BADRA2CADRA1AADRA1B
SCHEMBL1637444 0.83 ADRA2A (0.49) ADRA2AADRA2BADRA2CADRA1AADRA1B
SCHEMBL3070530 0.83 ADRA2A (0.51) ADRA2AADRA2BADRA2CADRA1AADRA1B
SCHEMBL3062104 0.82 ADRA2A (0.48) ADRA2AADRA2BADRA2CADRA1AADRA1B
SCHEMBL13089105 0.79 MAPT (0.38) ADRA2AADRA2BADRA1AADRA1DCYP2D6
SCHEMBL13247020 0.78 CYP1A2 (0.40) ADRA2AADRA2BADRA2CADRA1AADRA1B
SCHEMBL3070706 0.78 HRH3 (0.46) ADRA2AADRA2BADRA2CADRA1AADRA1B
SCHEMBL3017476 0.77 ADRA2A (0.47) ADRA2AADRA2BADRA2CADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155715-B1 ((PHENYL)IMIDAZOLYL)METHYLHETEROARYL COMPOUNDS ALLERGAN INC (US) 2013-03-13 EP disclosed
EP-2155715-A1 ((PHENYL)IMIDAZOLYL)METHYLHETEROARYL COMPOUNDS ALLERGAN, INC. (US) 2010-02-24 EP disclosed
WO-2008141312-A1 ((PHENYL)IMIDAZOLYL)METHYLHETEROARYL COMPOUNDS ALLERGAN, INC. (US) 2008-11-20 WO disclosed