SCHEMBL3674264

SCHEMBL3674264

O=C(NC[C@H]1NC[C@@H]2CCC[C@@H]21)c1onc2ccccc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.37
CNR2 P34972 3/20 0.37
RAB9A P51151 3/20 0.36
NPC1 O15118 3/20 0.36
ALDH1A1 P00352 6/20 0.36
KDM4E B2RXH2 3/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
HPGD P15428 2/20 0.35
HSD17B10 Q99714 2/20 0.35
GAA P10253 2/20 0.35
GLA P06280 1/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
ESR2 Q92731 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
HTT P42858 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
RBP4 P02753 1/20 0.34
LMNA P02545 1/20 0.34
ROCK1 Q13464 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3668373 0.84 ROCK1 (0.35) CNR1CNR2RAB9ANPC1ALDH1A1
SCHEMBL496256 0.83 HIF1A (0.50) ROCK1HIF1A
SCHEMBL496264 0.77 MAPT (0.42) MAPTSMN1; SMN2LMNA
SCHEMBL3677156 0.72 HCRTR1 (0.40) RAB9ANPC1KDM4E
SCHEMBL496159 0.69 HTR4 (0.50) CNR1CNR2
SCHEMBL496329 0.67 HIF1A (0.43) HIF1A
SCHEMBL6170415 0.67 USP2 (0.49) RAB9ANPC1ALDH1A1KDM4EL3MBTL1
SCHEMBL18703328 0.64 IP6K1 (0.50) RAB9ANPC1ALDH1A1KDM4EGAA
SCHEMBL497068 0.64 HPGD (0.41) RAB9ANPC1ALDH1A1L3MBTL1HPGD
SCHEMBL496425 0.64 KDM4E (0.35) RAB9ANPC1ALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2164847-A1 3-AZA-BICYCLO[3.3.0]OCTANE COMPOUNDS Actelion Pharmaceuticals Ltd. (CH) 2010-03-24 EP disclosed
WO-2009004584-A1 3-AZA-BICYCLO[3.3.0]OCTANE COMPOUNDS ACTELION PHARMACEUTICALS LTD (CH) 2009-01-08 WO disclosed