SCHEMBL3674545

SCHEMBL3674545

CC1C[C@H]2CN(C(=O)OC(C)(C)C)[C@H](CNC(=O)c3onc4ccccc34)[C@H]2C1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACACB O00763 12/20 0.36
KDM4E B2RXH2 1/20 0.35
PKM P14618 1/20 0.35
ACACA Q13085 10/20 0.35
ACKR3 P25106 1/20 0.34
NAMPT P43490 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
FAP Q12884 1/20 0.32
SCD5 Q86SK9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3677156 0.87 HCRTR1 (0.40) ACACBKDM4EPKMACACAACKR3
SCHEMBL496419 0.86 HIF1A (0.38) KDM4EPKMACKR3
SCHEMBL3641052 0.83 ACKR3 (0.36) ACACBKDM4EPKMACACAACKR3
SCHEMBL496426 0.81 KDM4E (0.41) KDM4E
SCHEMBL2442561 0.81 KDM4E (0.41) KDM4E
SCHEMBL496277 0.81 TP53 (0.39) ACKR3
SCHEMBL496193 0.78 GAA (0.35) ACACBMEN1KMT2A
SCHEMBL3674486 0.75 HCRTR1 (0.50)
SCHEMBL496423 0.75 NR1H2 (0.34) NAMPT
SCHEMBL496719 0.75 HTR4 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2164847-A1 3-AZA-BICYCLO[3.3.0]OCTANE COMPOUNDS Actelion Pharmaceuticals Ltd. (CH) 2010-03-24 EP disclosed
WO-2009004584-A1 3-AZA-BICYCLO[3.3.0]OCTANE COMPOUNDS ACTELION PHARMACEUTICALS LTD (CH) 2009-01-08 WO disclosed