SCHEMBL3677005

SCHEMBL3677005

Clc1ccc(OCC2=NCCN2)cc1.c1ccc2cc(OCC3=NCCN3)ccc2c1

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 12/20 0.85
MAOA P21397 3/20 0.63
MAOB P27338 3/20 0.63
CYP2D6 P10635 2/20 0.52
NFKB1 P19838 1/20 0.52
TAAR1 Q96RJ0 1/20 0.52
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
MAPT P10636 1/20 0.50
KMT2A Q03164 1/20 0.50
HTR1A P08908 4/20 0.48
ADRA2A P08913 4/20 0.48
ADRA2B P18089 4/20 0.48
ADRA2C P18825 4/20 0.48
ADRA1A P35348 3/20 0.46
ADRA1D P25100 2/20 0.46
ADRA1B P35368 2/20 0.46
CYP1A2 P05177 1/20 0.45
THRB P10828 1/20 0.45
TSHR P16473 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3163676 0.92 NISCH (1.00) NISCHMAOAMAOBCYP2D6NFKB1
SCHEMBL3172922 0.88 NISCH (0.71) NISCHMAOAMAOBCYP2D6HTR1A
Hydrochloric Acid SCHEMBL11251146 0.86 NISCH (0.69) NISCHMAOAMAOBCYP2D6HTR1A
Hydrochloric Acid SCHEMBL11541553 0.82 NISCH (0.63) NISCHMAOAMAOBCYP2D6HTR1A
SCHEMBL3173653 0.80 NISCH (0.68) NISCHMAOAMAOBCYP2D6TAAR1
SCHEMBL546875 0.79 NISCH (1.00) NISCHMAOAMAOBCYP2D6TAAR1
Fenmetozole SCHEMBL30295426 0.78 NISCH (0.65) NISCHMAOAMAOBCYP2D6TAAR1
Fenmetozole SCHEMBL635495 0.78 NISCH (0.65) NISCHMAOAMAOBCYP2D6TAAR1
Hydrochloric Acid SCHEMBL11259967 0.77 NISCH (0.97) NISCHMAOAMAOBCYP2D6TAAR1
Fenmetozole SCHEMBL29913217 0.77 NISCH (0.63) NISCHMAOAMAOBCYP2D6TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2173720-A2 2-IMIDAZOLINES HAVING A GOOD AFFINITY TO THE TRACE AMINE ASSOCIATED RECEPTORS (TAARS) F. Hoffmann-Roche AG (CH) 2010-04-14 EP claimed
WO-2009003868-A2 2 -IMIDAZOLINES HAVING A GOOD AFFINITY TO THE TRACE AMINE ASSOCIATED RECEPTORS (TAARS) F. HOFFMANN-LA ROCHE AG (CH) 2009-01-08 WO claimed