SCHEMBL3682308

SCHEMBL3682308

O=C(O)c1cc(-c2ccc(Cl)c(Cl)c2)[nH]n1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMO O15229 6/20 0.55
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
MAPT P10636 2/20 0.48
POLB P06746 1/20 0.48
NOTUM Q6P988 2/20 0.47
LDHA P00338 1/20 0.47
PPP1CA P62136 2/20 0.46
RPA1 P27694 2/20 0.44
KDM4E B2RXH2 1/20 0.44
USP2 O75604 1/20 0.44
GAA P10253 1/20 0.44
PKM P14618 1/20 0.44
ALOX12 P18054 1/20 0.44
HTT P42858 1/20 0.44
HCAR2 Q8TDS4 2/20 0.43
DAO P14920 1/20 0.43
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13883208 0.86 HCAR2 (0.47) KMOMEN1KMT2AMAPTPOLB
SCHEMBL1413913 0.83 NPC1 (0.55) KMOMEN1KMT2AMAPTPOLB
SCHEMBL8366435 0.82 NOTUM (0.57) MEN1KMT2AMAPTPOLBNOTUM
SCHEMBL31088355 0.82 NOTUM (0.57) MEN1KMT2AMAPTPOLBNOTUM
SCHEMBL13883211 0.80 HCAR2 (0.52) KMOMEN1KMT2AMAPTPOLB
SCHEMBL70360 0.80 CA12 (0.53) MEN1KMT2AMAPTPOLBHCAR2
SCHEMBL28168385 0.80 NOTUM (0.53) MEN1KMT2AMAPTNOTUMKDM4E
SCHEMBL14152313 0.79 HCAR2 (0.56) KMOMEN1KMT2AMAPTPOLB
SCHEMBL29019950 0.78 MEN1 (0.51) MEN1KMT2AMAPTPOLBHCAR2
SCHEMBL117667 0.78 MARS1 (0.60)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2167472-A2 1-BENZYLPYRAZOLE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF Sanofi-Aventis (FR) 2010-03-31 EP disclosed
WO-2009004171-A2 1-BENZYLPYRAZOLE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2009-01-08 WO disclosed