SCHEMBL3682377

SCHEMBL3682377

COc1ccc(OC)c(C=CC(=O)c2ccccc2NCCCN(C)C)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.56
PDE4B Q07343 1/20 0.56
PDE4C Q08493 1/20 0.56
PDE4D Q08499 1/20 0.56
ABCG2 Q9UNQ0 2/20 0.52
MAPT P10636 5/20 0.49
KDM4E B2RXH2 4/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
GAA P10253 3/20 0.49
ALDH1A1 P00352 3/20 0.49
HPGD P15428 3/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
POLB P06746 2/20 0.49
PAX8 Q06710 1/20 0.49
MCL1 Q07820 1/20 0.49
JUN P05412 1/20 0.49
NFKB1 P19838 1/20 0.49
LMNA P02545 2/20 0.47
ATM Q13315 2/20 0.47
NPSR1 Q6W5P4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3684125 0.95 PDE4A (0.57) PDE4APDE4BPDE4CPDE4DABCG2
SCHEMBL3694922 0.92 MAPT (0.57) PDE4APDE4BPDE4CPDE4DABCG2
SCHEMBL3682374 0.88 MAPT (0.56) PDE4APDE4BPDE4CPDE4DABCG2
SCHEMBL3687942 0.88 MAPT (0.56) PDE4APDE4BPDE4CPDE4DABCG2
SCHEMBL3688290 0.87 MAPT (0.58) PDE4APDE4BPDE4CPDE4DABCG2
SCHEMBL3697030 0.86 ABCG2 (0.59) PDE4APDE4BPDE4CPDE4DABCG2
SCHEMBL3694918 0.86 ABCG2 (0.59) PDE4APDE4BPDE4CPDE4DABCG2
SCHEMBL4851312 0.84 PDE4A (0.61) PDE4APDE4BPDE4CPDE4DABCG2
SCHEMBL3684123 0.83 MAPT (0.57) PDE4APDE4BPDE4CPDE4DABCG2
SCHEMBL3697931 0.83 MAPT (0.57) PDE4APDE4BPDE4CPDE4DABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US claimed
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed