SCHEMBL3684546

SCHEMBL3684546

OCCOc1cccc(CNCc2ccccc2)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 4/20 0.69
DRD4 P21917 2/20 0.60
DRD2 P14416 1/20 0.60
ADRA1D P25100 1/20 0.60
ADRA1A P35348 1/20 0.60
ADRA1B P35368 1/20 0.60
DRD3 P35462 1/20 0.60
ALDH1A1 P00352 3/20 0.56
RECQL P46063 1/20 0.56
SMN1; SMN2 Q16637 2/20 0.53
KDM4E B2RXH2 2/20 0.52
HTT P42858 1/20 0.52
CYP4F2 P78329 1/20 0.51
CYP4A11 Q02928 1/20 0.51
PPARG P37231 1/20 0.51
MAPK1 P28482 2/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
TDP1 Q9NUW8 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1037181 0.92 BCHE (0.67) BCHEDRD4DRD2ADRA1DADRA1A
SCHEMBL10809172 0.83 BCHE (0.67) BCHEDRD4DRD2ADRA1DADRA1A
SCHEMBL1240006 0.82 ALDH1A1 (0.48) BCHEDRD4DRD2ADRA1DADRA1A
SCHEMBL21634316 0.82 BCHE (0.63) BCHEDRD4DRD2ADRA1DADRA1A
SCHEMBL28545402 0.81 ALDH1A1 (0.62) BCHEDRD4DRD2ADRA1DADRA1A
SCHEMBL21634272 0.81 BCHE (0.67) BCHEDRD4DRD2ADRA1DADRA1A
SCHEMBL30821653 0.81 BCHE (0.67) BCHEDRD4DRD2ADRA1DADRA1A
SCHEMBL14724394 0.79 ALDH1A1 (0.57) DRD4DRD2ADRA1DADRA1AADRA1B
SCHEMBL30945670 0.79 HRH3 (0.45) MAPK1
SCHEMBL10011367 0.78 BCHE (0.76) BCHEALDH1A1KDM4ECYP4F2CYP4A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2185537-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS Pfizer Inc. (US) 2010-05-19 EP disclosed
WO-2009016498-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS PFIZER INC. (US) 2009-02-05 WO disclosed
WO-2009016498-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS PFIZER INC. (US) 2009-02-05 WO disclosed