SCHEMBL3686284

SCHEMBL3686284

Cc1csc(CN(C)C(=O)c2cc(C(N)=O)cc(N3CCCC3)c2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
KMT2A Q03164 1/20 0.40
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
NR1H4 Q96RI1 1/20 0.35
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
GAA P10253 1/20 0.33
KCNH2 Q12809 1/20 0.33
LOXL2 Q9Y4K0 2/20 0.32
USP2 O75604 1/20 0.32
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PIM1 P11309 2/20 0.32
PIM2 Q9P1W9 2/20 0.32
PIK3CA P42336 1/20 0.31
PIK3CB P42338 1/20 0.31
PRKD3 O94806 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3648036 0.84 RAB9A (0.42) KDM4EMEN1ALDH1A1KMT2ANPC1
SCHEMBL3351202 0.81 NPC1 (0.48) KDM4EMEN1ALDH1A1KMT2ANPC1
SCHEMBL3506848 0.81 RAB9A (0.40) KDM4EMEN1ALDH1A1KMT2ANPC1
SCHEMBL3511239 0.80 SLC5A7 (0.46) KDM4EALDH1A1NPC1RAB9AUSP2
SCHEMBL3509460 0.79 SLC5A7 (0.45) KDM4EALDH1A1NPC1RAB9ANR1H4
SCHEMBL3641877 0.79 NPC1 (0.41) KDM4EMEN1ALDH1A1KMT2ANPC1
SCHEMBL3509205 0.76 RAB9A (0.41) KDM4EMEN1ALDH1A1KMT2ANPC1
SCHEMBL3648778 0.75 MKNK1 (0.42) NPC1RAB9ALOXL2ALOX15
SCHEMBL166274 0.74 NPC1 (0.43) KDM4EMEN1ALDH1A1KMT2ANPC1
SCHEMBL3511235 0.73 IKBKB (0.36) KDM4EMEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2178837-A2 ISOPHTHALAMIDE DERIVATIVES INHIBITING BETA-SECRETASE ACTIVITY COMENTIS, INC. (US) 2010-04-28 EP disclosed
WO-2009015369-A2 COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2009-01-29 WO disclosed