SCHEMBL3686786

SCHEMBL3686786

CCCN(CCO)C(=O)c1cc([N+](=O)[O-])cc([N+](=O)[O-])c1N(CCOS(C)(=O)=O)CCOS(C)(=O)=O

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
HPGD P15428 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
TDP1 Q9NUW8 4/20 0.39
MAPK1 P28482 2/20 0.38
KDM4E B2RXH2 2/20 0.38
MAPT P10636 2/20 0.38
HKDC1 Q2TB90 1/20 0.37
HTT P42858 1/20 0.36
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
ALDH1A1 P00352 4/20 0.35
CHRNA7 P36544 1/20 0.33
TRPV1 Q8NER1 1/20 0.32
CYP19A1 P11511 1/20 0.32
HCAR3 P49019 2/20 0.32
POLB P06746 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3685725 0.95 KMT2A (0.41) KMT2AMEN1HPGDNPSR1TDP1
SCHEMBL3690192 0.95 KMT2A (0.41) KMT2AMEN1HPGDNPSR1TDP1
SCHEMBL3686404 0.89 KMT2A (0.42) KMT2AMEN1HPGDNPSR1TDP1
SCHEMBL3688122 0.89 KMT2A (0.42) KMT2AMEN1HPGDNPSR1TDP1
SCHEMBL3689649 0.85 KMT2A (0.46) KMT2AMEN1HPGDNPSR1TDP1
SCHEMBL3688111 0.85 KMT2A (0.45) KMT2AMEN1HPGDNPSR1TDP1
SCHEMBL3694331 0.84 KMT2A (0.50) KMT2AMEN1HPGDNPSR1TDP1
SCHEMBL3686829 0.84 KMT2A (0.50) KMT2AMEN1HPGDNPSR1TDP1
SCHEMBL3691401 0.84 KMT2A (0.50) KMT2AMEN1HPGDNPSR1TDP1
SCHEMBL3689656 0.83 KMT2A (0.40) KMT2AMEN1HPGDNPSR1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010044685-A1 NITROPHENYL MUSTARD ALCOHOLS, THEIR CORRESPONDING PHOSPHATES AND THEIR USE AS TARGETED CYTOTOXIC AGENTS AUCKLAND UNISERVICES LIMITED (NZ) 2010-04-22 WO claimed
WO-2010044685-A1 NITROPHENYL MUSTARD ALCOHOLS, THEIR CORRESPONDING PHOSPHATES AND THEIR USE AS TARGETED CYTOTOXIC AGENTS AUCKLAND UNISERVICES LIMITED (NZ) 2010-04-22 WO disclosed