SCHEMBL3687115

SCHEMBL3687115

COc1ccccc1-c1ccc(N2CCN(C)CC2)c(C(=O)C=Cc2ccc(O)cc2F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.45
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HIF1A Q16665 1/20 0.44
TUBB4A P04350 3/20 0.44
TUBB P07437 3/20 0.44
TUBA3C P0DPH7 3/20 0.44
TUBA1B P68363 3/20 0.44
TUBA4A P68366 3/20 0.44
TUBB4B P68371 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3686599 1.00 NR1H4 (0.45) NR1H4KDM4EMEN1ALDH1A1LMNA
SCHEMBL3686603 0.91 NR1H4 (0.47) NR1H4KDM4EMEN1ALDH1A1LMNA
SCHEMBL3695263 0.91 TUBB4A (0.45) KDM4EMEN1ALDH1A1LMNACYP1A2
SCHEMBL3694916 0.91 TUBB4A (0.45) KDM4EMEN1ALDH1A1LMNACYP1A2
SCHEMBL3697510 0.88 PTPN1 (0.43) KDM4EMEN1ALDH1A1LMNACYP1A2
SCHEMBL3693493 0.88 PTPN1 (0.43) KDM4EMEN1ALDH1A1LMNACYP1A2
SCHEMBL3688445 0.88 HDAC3 (0.51) ALDH1A1LMNASMN1; SMN2TUBB4ATUBB
SCHEMBL3689870 0.88 HDAC3 (0.51) ALDH1A1LMNASMN1; SMN2TUBB4ATUBB
SCHEMBL3690906 0.88 PTPN1 (0.48) KDM4EMEN1ALDH1A1LMNACYP1A2
SCHEMBL3697265 0.88 PTPN1 (0.48) KDM4EMEN1ALDH1A1LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US claimed
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed